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GPER1 gene

Known as: G protein-coupled estrogen receptor 1, G PROTEIN-COUPLED RECEPTOR 30, CEPR 
This gene plays a role in both estrogen binding and G protein-coupled receptor signaling.
National Institutes of Health

Related topics

Related topics

5 relations
G Protein-Coupled Receptor SignalingGPER protein, humanLigand BindingReceptor Signaling

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Review
2014
Review
2014
Estrogen biology: New insights into GPER function and clinical opportunities
Highly Cited
2011
Highly Cited
2011
Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity
Highly Cited
2010
Highly Cited
2010
Involvement of estrogen receptor variant ER-alpha36, not GPR30, in nongenomic estrogen signaling.
Accumulating evidence suggested that an orphan G protein-coupled receptor (GPR)30, mediates nongenomic responses to estrogen. The… 
Highly Cited
2009
Highly Cited
2009
In vivo Effects of a GPR30 Antagonist
Estrogen is central to many physiological processes throughout the human body. We have previously shown that the G protein… 
Highly Cited
2009
Highly Cited
2009
GPR30 Does Not Mediate Estrogenic Responses in Reproductive Organs in Mice
Abstract The G protein-coupled receptor Gpr30 (Gper) was recently claimed to bind to estradiol and to activate cytoplasmic signal… 
Highly Cited
2009
Highly Cited
2009
Chronic treatment with the G protein-coupled receptor 30 agonist G-1 decreases blood pressure in ovariectomized mRen2.Lewis rats.
The mRen2.Lewis congenic strain is an estrogen-sensitive model of hypertension whereby estrogen depletion produces a significant… 
Review
2008
Review
2008
The ins and outs of GPR30: A transmembrane estrogen receptor
Highly Cited
2006
Highly Cited
2006
17β-Estradiol, Genistein, and 4-Hydroxytamoxifen Induce the Proliferation of Thyroid Cancer Cells through the G Protein-Coupled Receptor GPR30
The higher incidence of thyroid carcinoma (TC) in women during reproductive years compared with men and the increased risk… 
Highly Cited
1998
Highly Cited
1998
Discovery of three novel G-protein-coupled receptor genes.
We report here the molecular cloning, tissue distribution, and chromosomal localization of novel genes encoding G-protein-coupled… 
Highly Cited
1996
Highly Cited
1996
Cloning of human cDNA encoding a novel heptahelix receptor expressed in Burkitt's lymphoma and widely distributed in brain and peripheral tissues.
Using PCR with degenerate primers and screening of a human B-cell lymphoblast cDNA library, a full-length cDNA encoding a 375… 
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