droloxifene

Known as: (E)--1-[4'-(2-dimethylaminoethyoxy)phenyl]-1(3-hydroxyphenyl)-2-phenyl-but-1-ene, (E)-3-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenyl-1-butenyl]phenol, 3-hydroxytamoxifen 
A phenolic analogue of tamoxifen, a nonsteroidal selective estrogen receptor modulator (SERM). Droloxifene competitively inhibits the binding of… (More)
National Institutes of Health

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1982-2014
051019822014

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2004
2004
OBJECTIVE The aim of this study was to evaluate the effect of conjugated equine oestrogen (CEE), and droloxifene, a selective… (More)
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2001
2001
Although increased levels of C-reactive protein have been linked to E therapy, the significance of this finding and whether it… (More)
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2001
2001
Human papillomavirus (HPV) type 16 infects the genital tract and is generally acknowledged to be a causative agent of cervical… (More)
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1998
1998
The identification and characterization of estrogen regulated genes in reproductive tissues is an important step in understanding… (More)
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1995
1995
The purpose of this study was to determine the effects of droloxifene (DRO), a new estrogen antagonist/agonist, on bone turnover… (More)
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1994
1994
Droloxifene, a new antiestrogen, has theoretical advantages over tamoxifen based on preclinical data. These include higher… (More)
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1992
1992
Droloxifene (3-OH-tamoxifen citrate) is a novel anti-oestrogen with a higher affinity for oestrogen receptors (ER), a lower… (More)
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1991
1991
Pharmacokinetics and metabolism of droloxifene, a new antiestrogenic drug, have been investigated by single- and multiple-dose… (More)
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1991
1991
We have previously shown that transforming growth factor beta (TGF beta) is a hormonally regulated negative growth factor in… (More)
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1989
1989
The effects of tamoxifen, three of its in vivo metabolites and 3-hydroxytamoxifen on cellular proliferation and the induction of… (More)
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