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setoperone

Known as: 5H-Thiazolo(3,2-a)pyrimidin-5-one, 6-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-2,3-dihydro-7-methyl- 
National Institutes of Health

Related topics

Related topics

4 relations

Broader (3)

Contrast MediaPyrimidinonesSerotonin Antagonists

Narrower (1)

fluorine-18-setoperone

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2012
2012
Positron emission tomography study of the effects of tryptophan depletion on brain serotonin(2) receptors in subjects recently remitted from major depression.
CONTEXT Decreased brain serotonin (5-hydroxytryptamine) levels are considered to mediate depressive relapse induced by the… 
2004
2004
Effect of serotonin antagonism in schizophrenia: A pilot study with setoperone
The new antipsychotic drug setoperone is pharmacologically characterized by its potent serotonin and moderate dopamine receptor… 
2004
2004
Risperidone (R 64 766), a potent and complete LSD antagonist in drug discrimination by rats
Risperidone was studied in a 0.16 mg/kg LSD-saline drug discrimination test procedure. At doses varying from 0.0025 to 0.63 mg/kg… 
Highly Cited
2000
Highly Cited
2000
A voxel-by-voxel analysis of [18F]setoperone PET data shows no substantial serotonin 5-HT2A receptor changes in schizophrenia
1999
1999
Relationship between central and peripheral serotonin 5-HT2A receptors: a positron emission tomography study in healthy individuals
Review
1996
Review
1996
Risperidone and related 5HT2/D2 antagonists: a new type of antipsychotic agent?
1989
1989
Activation of tuberoinfundibular dopamine neurons following the acute administration of atypical antipsychotics.
Highly Cited
1988
Highly Cited
1988
Antagonism of serotonin receptor mediated neuroendocrine and temperature responses by atypical neuroleptics in the rat.
1988
1988
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
LY53857, spiperone, ketanserin, and setoperone were potent and competitive 5-HT2-receptor antagonists in the rat jugular vein… 
1987
1987
Opposite regulation of serotonin-S2 and dopamine-D2 receptors in rat brain following chronic receptor blockade.
Rats were chronically treated with setoperone, a mixed serotonin and dopamine antagonist. Alterations in serotonin-S2 and… 
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