Skip to search formSkip to main contentSkip to account menu

setoperone

Known as: 5H-Thiazolo(3,2-a)pyrimidin-5-one, 6-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-2,3-dihydro-7-methyl- 
National Institutes of Health

Related topics

Related topics

4 relations

Broader (3)

Contrast MediaPyrimidinonesSerotonin Antagonists

Narrower (1)

fluorine-18-setoperone

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2004
2004
Effects of 5-HT1A agonists and 5-HT2 antagonists on haloperidol-induced dyskinesias in squirrel monkeys: no evidence for reciprocal 5-HT-dopamine interaction
Dyskinetic movements and dystonic postures may be induced by neuroleptics in monkeys that have undergone previous neuroleptic… 
Highly Cited
2000
Highly Cited
2000
A voxel-by-voxel analysis of [18F]setoperone PET data shows no substantial serotonin 5-HT2A receptor changes in schizophrenia
Review
1996
Review
1996
Risperidone and related 5HT2/D2 antagonists: a new type of antipsychotic agent?
1995
1995
Pet imaging of human pituitary 5-HT2 receptors with F-18 setoperone
Serotonin (5-HT) receptors play an important role in the regulation of pituitary function. In particular, 5HT agonists stimulate… 
1990
1990
[Development of new antipsychotic drugs].
As far as schizophrenia is concerned, therapeutical effects of neuroleptics based on brain-located dopamine receptor blockers are… 
1989
1989
Activation of tuberoinfundibular dopamine neurons following the acute administration of atypical antipsychotics.
1988
1988
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
LY53857, spiperone, ketanserin, and setoperone were potent and competitive 5-HT2-receptor antagonists in the rat jugular vein… 
1988
1988
Dopamine neurochemical profile of atypical antipsychotics resembles that of D-1 antagonists
SummaryThe release and metabolism of dopamine in the mouse caudate-putamen were determined after the oral administration of… 
Review
1988
Review
1988
Receptor interactions of dopamine and serotonin antagonists: binding in vitro and in vivo and receptor regulation.
The advent of receptor binding techniques has provided new ways of studying the mechanism of action of drugs. In vitro… 
1986
1986
Neuroendocrine effects of setoperone: a new neuroleptic drug.
Setoperone (R 52245), a serotonin S2 and dopamine D2 receptor blocker, was tested on eight healthy male volunteers, receiving 5… 
By clicking accept or continuing to use the site, you agree to the terms outlined in our Privacy Policy (opens in a new tab), Terms of Service (opens in a new tab), and Dataset License (opens in a new tab)