imidazobenzodiazepine

Alcohol (ethanol, EtOH) has pleiotropic actions and induces a number of acute and long‐term effects due to direct actions on… Expand

Several structural subclasses of ligands bind to the benzodiazepine (BZD) binding site of the GABA(A) receptor. Previous studies… Expand

We characterized modulation of the gamma-aminobutyric acid (GABA)-evoked responses of the diazepam-insensitive alpha 4 beta 2… Expand

Flumazenil, an imidazobenzodiazpine, is the first benzodiazepine antagonist available for clinical use. It is a specific… Expand

Abstract: Ro 15‐4513 (ethyl‐8‐azido‐5,6‐dihydro‐5‐methyl‐6‐oxo‐4H‐imidazo[1,5‐a][1,4]benzodiazepine‐3‐carboxylate), a partial… Expand

The imidazobenzodiazepine, Ro15-4513, which is a partial inverse agonist at brain benzodiazepine receptors, reversed the… Expand

Ethanol, at pharmacologically relevant concentrations of 20 to 100 mM, stimulates gamma-aminobutyric (GABA) receptor-mediated… Expand

Midazolam is an imidazobenzodiazepine with unique properties when compared with other benzodiazepines. It is water soluble in its… Expand

Le midazolam est au moins aussi efficace que le diazepam, les malades le preferent en general; il y a moins de complications… Expand

Abstract The imidazobenzodiazepine RO 15-1788 is a specific proconvulsant against isoniazid induced convulsions when given… Expand