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CB 3717
Known as:
CB-3717
, CB3717
National Institutes of Health
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Related topics
Related topics
6 relations
Broader (5)
Antineoplastic Agents
Enzyme Inhibitors
Folic Acid
Folic Acid Antagonists
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analogs & derivatives
Papers overview
Semantic Scholar uses AI to extract papers important to this topic.
2012
2012
Abstract 1929: Antifolates as folate receptor targeting ligands: Design and synthesis of their conjugates with cytotoxic agents
I. Vlahov
,
Fei You
,
Ryan Dorton
,
Elaine Westrick
,
J. Reddy
,
C. Leamon
2012
Corpus ID: 56874626
Proceedings: AACR 103rd Annual Meeting 2012‐‐ Mar 31‐Apr 4, 2012; Chicago, IL Antifolates are interfering specifically with DNA…
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2006
2006
DNA Damage and p 53 Induction Do Not Cause ZD 1694-induced Cell Cycle Arrest in Human Colon Carcinoma Cells '
Sei-ichi
,
Matsui
,
+6 authors
Rustum
2006
Corpus ID: 17498289
Using four complementary approaches, i.e., cell synchronization, bro modeoxyuridlne labeling, and DNA and Western blot analyses…
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1988
1988
PHARMACOKINETIC AND TOXICITY STUDIES WITH C2-DESAMINO-C2-SUBSTITUTED ANALOGS OF THE ANTIFOLATE N10-PROPARGYL-5,8-DIDEAZAFOLIC ACID (CB3717)
Newell
,
R. Maxwell
,
Griffiths
,
G. M. F. Bisset
,
L. Hughes
,
A. Calvert
1988
Corpus ID: 63768946
1988
1988
2-DESAMINO-2-SUBSTITUTED ANALOGS OF 10-PROPARGYL-5,8-DEAZAFOLATE (CB3717) AS INHIBITORS OF THYMIDYLATE SYNTHASE (TS)
J. Bishop
,
A. Jackman
,
L. Hughes
,
P. Marsham
,
T. Jones
,
A. Calvert
1988
Corpus ID: 68097420
1987
1987
POLYGLUTAMATION OF THE THYMIDYLATE SYNTHASE (TS) INHIBITOR N-10-PROPARGYL-5,8-DIDEAZAFOLIC ACID (CB3717) IN L1210 CELLS-INVITRO
E. Sikora
,
A. Jackman
,
Newell
,
A. Calvert
1987
Corpus ID: 74708583
Review
1987
Review
1987
A REVIEW OF THE DEVELOPMENT OF N-10-PROPARGYL-5,8-DIDEAZAFOLIC ACID (CB3717)
A. Calvert
1987
Corpus ID: 68418405
1984
1984
EARLY CLINICAL-STUDIES WITH CB3717 ((N-(4-(N-(2-AMINO-4-HYDROXY-6-QUINAZOLINYL)METHYL)PROP-2-YNYLAMINO)BENZOYL)-L-GLUTAMIC ACID
A. Calvert
,
D. Alison
,
+5 authors
K. R. Harrap
1984
Corpus ID: 62316705
1984
1984
STUDIES ON THE MECHANISM OF CB3717 INDUCED HEPATOTOXICITY
Newell
,
D. Alison
,
A. Jackman
,
A. Calvert
,
K. Harrap
1984
Corpus ID: 74603161
1983
1983
PHASE-I STUDIES WITH CB3717 (N-(4-(N-AMINO-4-HYDROXY-6-QUINAZOLINLY)METHYL)PROP-2-YNYLAMINO)BENZOYL)-L-GLUTAMIC ACID)
A. Calvert
,
D. Alison
,
+4 authors
K. R. Harrap
1983
Corpus ID: 78647691
1983
1983
TOXICITY AND PHARMACOKINETIC STUDIES WITH CB3717
Newell
,
Z. Siddik
,
+5 authors
K. Harrap
1983
Corpus ID: 74692887