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picrotoxinin

Known as: (1aR-(1a alpha,2a beta,3 beta,6 beta,6a beta,8aS*,8b beta,9R*))-hexahydro-2a-hydroxy-8b-methyl-9-(1-methylethenyl)-3,6-methano-8H-1,5,7-trioxa cyclopenta(ij)cycloprop(a)azulene-4,8(3H)-dione, picrotoxinine 
National Institutes of Health

Related topics

Related topics

3 relations

Broader (2)

GABA-A Receptor AntagonistsPicrotoxin
analogs & derivatives

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Review
2005
Review
2005
GABA(A) receptor channel pharmacology.
  • G. Johnston
  • Current pharmaceutical design
  • 2005
  • Corpus ID: 11911600
GABA(A) receptor channels are ubiquitous in the mammalian central nervous system mediating fast inhibitory neurotransmission by… 
Highly Cited
2004
Highly Cited
2004
The human taste receptor hTAS2R14 responds to a variety of different bitter compounds.
Highly Cited
2001
Highly Cited
2001
Effects of membrane cholesterol on the sensitivity of the GABAA receptor to GABA in acutely dissociated rat hippocampal neurones
Highly Cited
2001
Highly Cited
2001
GLC‐3: a novel fipronil and BIDN‐sensitive, but picrotoxinin‐insensitive, L‐glutamate‐gated chloride channel subunit from Caenorhabditis elegans
We report the cloning and expression of a novel Caenorhabditis elegans polypeptide, GLC‐3, with high sequence identity to… 
Review
1997
Review
1997
Molecular biology of insect neuronal GABA receptors
Highly Cited
1994
Highly Cited
1994
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
Highly Cited
1994
Highly Cited
1994
N-containing sugars from Morus alba and their glycosidase inhibitory activities.
Highly Cited
1993
Highly Cited
1993
A point mutation in a Drosophila GABA receptor confers insecticide resistance
VERTEBRATES and invertebrates both have GABA (γ-aminobutyric acid) as a major inhibitory neurotransmitter1,2. GABAA receptors in… 
Highly Cited
1992
Highly Cited
1992
The atypical M2 segment of the beta subunit confers picrotoxinin resistance to inhibitory glycine receptor channels.
Purified preparations of the inhibitory glycine receptor (GlyR) contain alpha and beta subunits, which share homologous primary… 
Highly Cited
1978
Highly Cited
1978
Interaction of barbiturates with dihydropicrotoxinin binding sites related to the GABA receptor-ionophore system.
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