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normetazocine

Known as: 1,2,3,4,5,6-hexahydro-6,11-dimethyl-2,6-methano-3-benzazocin-8-ol, norcyclazocine 
National Institutes of Health

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2 relations

Broader (1)

Cyclazocine
analogs & derivatives

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2018
2018
Synthesis and Structure-Activity Relationships of LP1 Derivatives: N-Methyl-N-phenylethylamino Analogues as Novel MOR Agonists
The opioid pharmacological profile of cis-(−)-N-normetazocine derivatives is deeply affected by the nature of their N… 
2008
2008
The influence of esters and carboxylic acids as the N-substituent of opioids. Part 1: Benzomorphans.
2002
2002
Synthesis and pharmacological evaluation of 6-piperidino- and 6-piperazinoalkyl-2(3H)-benzothiazolones as mixed sigma/5-HT(1A) ligands.
1997
1997
Synthesis of (+)-(1'R,2'S) and (1'S,2'R)-6,11-dimethyl-1,2,3,4,5,6 -hexahydro-3-[[2'-(alkoxycarbonyl)-2'-phenylcyclopropyl]methyl]-2 ,6 -methano-3-benzazocin-8-ol. Comparison of the affinities for…
The synthesis and the in vitro receptor affinity for sigma 1 and opiod receptors of the two diastereoisomers of (+)-cis-MPCB… 
1991
1991
Electrophilic gamma-lactone kappa-opioid receptor probes. Analogues of 2'-hydroxy-2-tetrahydrofurfuryl-5,9-dimethyl-6,7-benzomorphan diastereomers.
Benzomorphans with an electrophilic group in the nitrogen substituent were prepared as potentially irreversible ligands for the… 
1985
1985
Synthesis of some N-substituted 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines (6,7-benzomorphans).
In order to study the effects of N-substituents of benzomorphans on antagonist-agonist activity we synthesized several… 
1980
1980
Synthesis and biological activity of fluoroalkylamine derivatives of narcotic analgesics.
N-Ethyl-, N-(2-fluoroethyl)-, N-(2,2-difluoroethyl)-, and N-(2,2,2-trifluoroethyl)-substituted normeperidine (1b-e) and… 
1977
1977
N-(2,4,5-Trihydroxyphenehtyl)normetazocine, a potential irreversible inhibitor of the narcotic receptor.
The reaction of N-2,4,5-tribenzyloxyphenyl)ethyl methanesulfonate, prepared in a seven-step sequence, with normetazocine followed… 
1977
1977
Potential long acting opiate antagonists: preparation, pharmacological activity, and opiate-receptor binding of N-substituted 2'-hydroxy-5-methyl-9 alpha-propyl-6,7-benzomorphans.
A homologous series of N-substituted 2'-hydroxy-5-methyl-9 alpha-propyl-6,7-benzomorphans (hydrogen to octyl inclusive, allyl… 
1974
1974
The quantitation of cyclazocine and its metabolites in human urine by use of gas-liquid chromatography.
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