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Cyclazocine

Known as: 2,6-Methano-3-benzazocin-8-ol, 3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-, Cyclazocine [Chemical/Ingredient] 
An analgesic with mixed narcotic agonist-antagonist properties.
National Institutes of Health

Papers overview

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Highly Cited
1995
Highly Cited
1995
The ability of mu-opioid agonists to activate G proteins has been demonstrated by studying the binding of the GTP analogue… Expand
Highly Cited
1988
Highly Cited
1988
Abstract: The potent noncompetitive N‐methyl‐D‐aspartate (NMDA) receptor antagonist [3H]MK‐801 bound with nanomolar affinity to… Expand
Highly Cited
1986
Highly Cited
1986
The kappa opioid agonists are analgesics that seem to be free of undesired morphine-like effects. Their dysphoric actions… Expand
Highly Cited
1982
Highly Cited
1982
  • T. Su
  • The Journal of pharmacology and experimental…
  • 1982
  • Corpus ID: 23837713
A portion of the specific binding of tritiated SKF-10047 to the guinea-pig brain suspension of the particulate fraction is not… Expand
Highly Cited
1976
Highly Cited
1976
A series of morphine-like and nalorphine-like drugs were studied in the nondependent, morphine-dependent and cyclazocine… Expand
Highly Cited
1975
Highly Cited
1975
1 Morphine inhibits the electrically evoked (0.1‐0.15 Hz, 1 ms) contractions of the longitudinal muscle of the mouse vas deferens… Expand
Highly Cited
1975
Highly Cited
1975
The analgesic activity of morphine and the narcotic antagonists, pentazocine, cyclazocine, levallorphan and nalorphine, was… Expand
Highly Cited
1973
Highly Cited
1973
Naltrexone (EN-1639A) is approximately 17 times more potent than nalorphine as an antagonist in man. It is virtually devoid of… Expand
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Highly Cited
1966
Highly Cited
1966
The potent narcotic antagonist, cyclazocine, has a long duration of action and is effective when administered orally. Although… Expand
Highly Cited
1965
Highly Cited
1965
The effects of single doses and chronic administration of cyclazocine have been studied in nontolerant postaddicts, as well as in… Expand