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Cyclazocine

Known as: 2,6-Methano-3-benzazocin-8-ol, 3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-, Cyclazocine [Chemical/Ingredient] 
An analgesic with mixed narcotic agonist-antagonist properties.
National Institutes of Health

Papers overview

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Highly Cited
1998
Highly Cited
1998
There is accumulating evidence that kappa opioid agonists attenuate cocaine's behavioral effects, and we recently reported that… Expand
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Highly Cited
1996
Highly Cited
1996
In C6 glioma cells stably expressing a homogeneous population of the cloned rat mu opioid receptor, the binding affinities of… Expand
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Highly Cited
1995
Highly Cited
1995
The ability of mu-opioid agonists to activate G proteins has been demonstrated by studying the binding of the GTP analogue… Expand
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Highly Cited
1986
Highly Cited
1986
The kappa opioid agonists are analgesics that seem to be free of undesired morphine-like effects. Their dysphoric actions… Expand
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1986
1986
The activity of ketocyclazocine, a putative kappa opioid receptor agonist, was studied and compared with that of morphine, a mu… Expand
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Highly Cited
1982
Highly Cited
1982
  • T. P. Su
  • The Journal of pharmacology and experimental…
  • 1982
  • Corpus ID: 23837713
A portion of the specific binding of tritiated SKF-10047 to the guinea-pig brain suspension of the particulate fraction is not… Expand
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Highly Cited
1976
Highly Cited
1976
A series of morphine-like and nalorphine-like drugs were studied in the nondependent, morphine-dependent and cyclazocine… Expand
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1976
1976
Rats were trained to press a lever in order to stimulate their lateral hypothalamus through a chronically implanted electrode… Expand
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Highly Cited
1975
Highly Cited
1975
The analgesic activity of morphine and the narcotic antagonists, pentazocine, cyclazocine, levallorphan and nalorphine, was… Expand
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Highly Cited
1973
Highly Cited
1973
Naltrexone (EN-1639A) is approximately 17 times more potent than nalorphine as an antagonist in man. It is virtually devoid of… Expand
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