carebastine

Known as: Benzeneacetic acid, 4-(4-(4-(diphenylmethoxy)-1-piperidinyl)-1-oxobutyl)-alpha,alpha-dimethyl- 
 
National Institutes of Health

Topic mentions per year

Topic mentions per year

1988-2014
02419882014

Papers overview

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2009
2009
Ebastine is a well-known selective second-generation histamine H(1) receptor antagonist, which is used for seasonal and perennial… (More)
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2006
2006
Ebastine undergoes extensive metabolism to form desalkylebastine and hydroxyebastine. Hydroxyebastine is subsequently metabolized… (More)
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2004
2004
The oxidation of tert-butyl-phenyl group of title compounds by some microorganisms was studied. We have optimized the conditions… (More)
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2001
2001
Ebastine (CAS 90729-43-4) is an antiallergic agent which selectively and potently blocks histamine H1-receptors in vivo. A simple… (More)
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2001
2001
AIMS Sedation induced by antihistamines is widely recognized to be caused by their penetration through the blood-brain-barrier… (More)
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2000
2000
The transport mechanism of the non-sedative H1-antagonist ebastine and its first-pass carboxylic acid metabolite carebastine at… (More)
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Review
2000
Review
2000
  • P Kingham
  • Current opinion in investigational drugs
  • 2000
Carebastine, a histamine H1 antagonist, is under development by Almirall Prodesfarma for the potential treatment of allergic… (More)
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1994
1994
Pharmacokinetics of ebastine (CAS 90729-43-4), a histamine H1-receptor antagonist, was evaluated in healthy male volunteers. The… (More)
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1994
1994
The pharmacokinetics of ebastine (CAS 90729-43-4), a new histamine H1-receptor antagonist, was investigated in rats, guinea pigs… (More)
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1993
1993
Ebastine is an H1-receptor antagonist with a relative lack of sedating properties. It is almost completely converted to… (More)
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