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Histamine H1 Antagonists

Known as: Antagonists, Histamine H1, H1 Antagonists, Histamine, Antihistaminics, H1 
Drugs that selectively bind to but do not activate histamine H1 receptors, thereby blocking the actions of endogenous histamine. Included here are… Expand
National Institutes of Health

Related topics

Related topics

49 relations

Narrower (40)

AntazolineAzelastine hydrochlorideCinnarizineClemastine
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Anti-Allergic AgentsBronchodilator AgentsHypnotics and SedativesImmediate hypersensitivity
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Broader (2)

AntihistaminesHistamine Antagonists

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Highly Cited
2011
Highly Cited
2011
Structure of the human histamine H1 receptor complex with doxepin
The biogenic amine histamine is an important pharmacological mediator involved in pathophysiological processes such as allergies… Expand
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Highly Cited
2007
Highly Cited
2007
A Pseudo-Response Regulator is misexpressed in the photoperiod insensitive Ppd-D1a mutant of wheat (Triticum aestivum L.)
Ppd-D1 on chromosome 2D is the major photoperiod response locus in hexaploid wheat (Triticum aestivum). A semi-dominant mutation… Expand
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Highly Cited
2005
Highly Cited
2005
The Pseudo-Response Regulator Ppd-H1 Provides Adaptation to Photoperiod in Barley
Plants commonly use photoperiod (day length) to control the timing of flowering during the year, and variation in photoperiod… Expand
Highly Cited
2004
Highly Cited
2004
Human SirT1 interacts with histone H1 and promotes formation of facultative heterochromatin.
We characterized human SirT1, one of the human homologs of the budding yeast Sir2p, an NAD+-dependent histone deacetylase… Expand
Highly Cited
2002
Highly Cited
2002
Nucleotide exchange factor GEF-H1 mediates cross-talk between microtubules and the actin cytoskeleton
Regulation of the actin cytoskeleton by microtubules is mediated by the Rho family GTPases. However, the molecular mechanisms… Expand
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Highly Cited
2000
Highly Cited
2000
Dynamic binding of histone H1 to chromatin in living cells
The linker histone H1 is believed to be involved in chromatin organization by stabilizing higher-order chromatin structure… Expand
Highly Cited
1999
Highly Cited
1999
OATP and P-glycoprotein transporters mediate the cellular uptake and excretion of fexofenadine.
Fexofenadine, a nonsedating antihistamine, does not undergo significant metabolic biotransformation. Accordingly, it was… Expand
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Highly Cited
1995
Highly Cited
1995
Human immunodeficiency virus type 1 viral protein R (Vpr) arrests cells in the G2 phase of the cell cycle by inhibiting p34cdc2 activity.
The Vpr accessory gene product of human immunodeficiency virus types 1 and 2 and simian immunodeficiency virus is believed to… Expand
Highly Cited
1994
Highly Cited
1994
Inhibition of cyclin-dependent kinases by purine analogues.
While testing purines related to the non-specific protein kinase inhibitors N6-dimethylaminopurine and N6-(delta 2-isopentenyl… Expand
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Highly Cited
1988
Highly Cited
1988
Drugs abused by humans preferentially increase synaptic dopamine concentrations in the mesolimbic system of freely moving rats.
The effect of various drugs on the extracellular concentration of dopamine in two terminal dopaminergic areas, the nucleus… Expand
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