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altanserin

Known as: 3-(2-(4-(p-Fluorobenzoyl)piperidino)ethyl)-2-thio-2,4(1H,3H)-quinazolinedione, R 53200, 4(1H)-Quinazolinone, 3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-2,3-dihydro-2-thioxo- 
 
National Institutes of Health

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5 relations

Broader (3)

Contrast MediaKetanserinSerotonin Antagonists
altanserin tartrateanalogs & derivatives

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2016
2016
Serotonin 2A receptor agonist binding in the human brain with [11C]Cimbi-36: Test–retest reproducibility and head-to-head comparison with the antagonist [18F]altanserin
INTRODUCTION [(11)C]Cimbi-36 is a recently developed serotonin 2A (5-HT2A) receptor agonist positron emission tomography (PET… Expand
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Highly Cited
2010
Highly Cited
2010
Decreased frontal serotonin2A receptor binding in antipsychotic-naive patients with first-episode schizophrenia.
CONTEXT Postmortem investigations and the receptor affinity profile of atypical antipsychotics have implicated the participation… Expand
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2005
2005
Binding characteristics of the 5-HT2A receptor antagonists altanserin and MDL 100907.
To study the 5-HT(2A) receptors in the living human brain, using positron emission tomography (PET), two selective radiotracers… Expand
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2003
2003
Influence of synaptic serotonin level on [18F]altanserin binding to 5HT2 receptors in man
The feasibility of in vivo serotonin 5HT(2) receptor binding measurement using [18F]altanserin as a radioligand has been well… Expand
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2001
2001
Analyses of [(18)F] altanserin bolus injection PET data. I: consideration of radiolabeled metabolites in baboons.
Positron emission tomography (PET) has been used to study serotonin 2A (5-HT(2A)) receptor binding in human brain using the 5-HT… Expand
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1999
1999
Characterization of radioactive metabolites of 5-HT2A receptor PET ligand [18F]altanserin in human and rodent.
This study was performed to identify and characterize the radiometabolites of the serotonin 5-HT2A receptor ligand [18F… Expand
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Highly Cited
1996
Highly Cited
1996
Sex difference in 5HT2 receptor in the living human brain
Serotonergic mechanisms are involved in gender-related behaviors and psychiatric conditions like aggression, eating disorders… Expand
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1995
1995
Serotonin 5HT2 Receptor Imaging in the Human Brain Using Positron Emission Tomography and a New Radioligand, [18F]Altanserin: Results in Young Normal Controls
Changes in serotonin-2 receptors have been demonstrated in brain autopsy material from patients with various neurodegenerative… Expand
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Highly Cited
1995
Highly Cited
1995
Serotonergic modulation of striatal dopamine measured with positron emission tomography (PET) and in vivo microdialysis
Positron emission tomography and in vivo microdialysis were used to study serotonin's role in modulating striatal dopamine… Expand
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Highly Cited
1987
Highly Cited
1987
Stimulation of corticosterone and beta-endorphin secretion in the rat by selective 5-HT receptor subtype activation.
Changes in plasma concentrations of corticosterone and beta-endorphin (beta-END) were determined in male rats after treatment… Expand
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