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Sumatriptan

Known as: 1-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-N-methyl-methanesulfonamide, Sumatriptán, 3-(2-(Dimethylamino)ethyl)-N-methyl-1H-indole-5-methanesulfonamide 
A sulfonamide triptan with vasoconstrictor activity. Sumatriptan selectively binds to and activates serotonin 5-HT1D receptors in the central nervous… 
National Institutes of Health

Related topics

Related topics

43 relations
0.5 ML Sumatriptan 12 MG/ML Cartridge0.5 ML Sumatriptan 12 MG/ML Cartridge [Imitrex]0.5 ML Sumatriptan 12 MG/ML Jet Injector [Sumavel]0.5 ML Sumatriptan 12 MG/ML Prefilled Syringe

Narrower (10)

AlsumaCP 122288CP 122638GR-43175

Broader (5)

Serotonin 5-HT1 Receptor AgonistsSulfonamidesTriptansVasoconstrictor Agents

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2003
2003
Impact of a Group‐Based Model of Disease Management for Headache
Objectives.—To assess the impact of a group‐based model of disease management for patients with headache. 
Review
2002
Review
2002
Integrating the triptans into clinical practice
&NA; The triptans (selective serotonin agonists) are becoming the first‐line alternatives in the acute pharmacological treatment… 
Review
2000
Review
2000
Eletriptan in acute migraine: a double-blind, placebo-controlled comparison to sumatriptan.
5. Spierings ELH. Therapeutic gain: a critique. Headache 1999;39:517– 518. Letter. 6. Tfelt-Hansen P, Teall J, Rodriguez F, et al… 
Highly Cited
2000
Highly Cited
2000
Desensitisation of 5-HT autoreceptors upon pharmacokinetically monitored chronic treatment with citalopram.
2000
2000
Autoradiography of receptor-activated G-proteins in post mortem human brain
Review
1999
Review
1999
Pharmacological aspects of experimental headache models in relation to acute antimigraine therapy.
Highly Cited
1998
Highly Cited
1998
Selective labelling of 5-HT7 receptor recognition sites in rat brain using [3H]5-carboxamidotryptamine
Highly Cited
1998
Highly Cited
1998
The canine external carotid vasoconstrictor 5-HT1 receptor: blockade by 5-HT1B (SB224289), but not by 5-HT1D (BRL15572) receptor antagonists.
Highly Cited
1995
Highly Cited
1995
[3H]sumatriptan labels both 5-HT1D and 5-HT1F receptor binding sites in the guinea pig brain: an autoradiographic study
We have used in vitro autoradiography to visualize [3H]sumatriptan binding sites in sections of guinea-pig and rat brain. In… 
Review
1995
Review
1995
Presynaptic 5-HT auto- and heteroreceptors in the human central and peripheral nervous system
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