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CP 122288

Known as: 1H-Indole-5-methanesulfonamide, N-methyl-3-((1-methyl-2-pyrrolidinyl)methyl)-, (R)-, CP-122,288, CP-122288 
National Institutes of Health

Related topics

Related topics

3 relations

Broader (2)

PyrrolidinesSumatriptan
analogs & derivatives

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2001
2001
pH‐Mediated field‐amplified sample stacking of pharmaceutical cations in high‐ionic strength samples
Capillary electrophoretic separation of samples of physiological origin typically have both poor resolution and efficiency due to… 
Highly Cited
2000
Highly Cited
2000
No acute antimigraine efficacy of CP‐122,288, a highly potent inhibitor of neurogenic inflammation: Results of two randomized, double‐blind, placebo‐controlled clinical trials
CP‐122,288 is a highly potent inhibitor of neurogenic plasma extravasation in animal models at doses without vasoconstrictor… 
1998
1998
Human 5-HT1F receptor-stimulated [35S]GTPgammaS binding: correlation with inhibition of guinea pig dural plasma protein extravasation.
1997
1997
The 5-HT1D Receptor Antagonist GR-127,935 Prevents Inhibitory Effects of Sumatriptan but not CP-122,288 and 5-CT on Neurogenic Plasma Extravasation within Guinea Pig Dura Mater
Highly Cited
1995
Highly Cited
1995
Autoradiographic visualisation of [3H]5-carboxamidotryptamine binding sites in the guinea pig and rat brain.
Highly Cited
1995
Highly Cited
1995
[3H]sumatriptan labels both 5-HT1D and 5-HT1F receptor binding sites in the guinea pig brain: an autoradiographic study
We have used in vitro autoradiography to visualize [3H]sumatriptan binding sites in sections of guinea-pig and rat brain. In… 
1995
1995
The in vivo pharmacological profile of a 5‐HT1 receptor agonist, CP‐122, 288, a selective inhibitor of neurogenic inflammation
1 The aim of the present study was to investigate the in vivo pharmacological profile of CP‐122, 288, an indole‐derivative with a… 
1995
1995
Suppression by the sumatriptan analogue, CP‐122,288 of c‐fos immunoreactivity in trigeminal nucleus caudalis induced by intracisternal capsaicin
1 The effects of an intravenously administered sumatriptan analogue were examined on c‐fos‐like immunoreactivity (c‐fos‐LI), a… 
1995
1995
The pre- and postjunctional activity of CP-122,288, a conformationally restricted analogue of sumatriptan.
1995
1995
Effect of a 5‐HT1 receptor agonist, CP‐122,288, on oedema formation induced by stimulation of the rat saphenous nerve
Neurogenic oedema formation in the rat hind paw skin induced by electrical stimulation of the saphenous nerve and measured by… 
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