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Metribolone

Known as: 17 beta-Hydroxy-17 alpha-methylestra-4,9,11-trien-3-one, Metribolone [Chemical/Ingredient], Methyltrienolone 
A synthetic non-aromatizable androgen and anabolic steroid. It binds strongly to the androgen receptor and has therefore also been used as an… 
National Institutes of Health

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In Bloodagonistsanalogs & derivativesantagonists & inhibitors

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R-1881

Papers overview

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2012
2012
Androgens and estrogens prevent rosiglitazone-induced adipogenesis in human mesenchymal stem cells
Thiazolidinediones (TZD), a class of anti-diabetic drugs, determine bone loss and increase fractures particularly in post… 
Highly Cited
1995
Highly Cited
1995
Abnormal androgen receptor binding affinity in subjects with Kennedy's disease (spinal and bulbar muscular atrophy).
We have investigated androgen-binding properties of the androgen receptor (AR) in cultured suprapubic skin fibroblasts from six… 
Highly Cited
1988
Highly Cited
1988
A high abundance androgen receptor in goldfish brain: characteristics and seasonal changes.
Testosterone (T) exerts its actions in brain directly via androgen receptors or, after aromatization to estradiol, via estrogen… 
Highly Cited
1985
Highly Cited
1985
Mechanism of androgen-receptor augmentation. Analysis of receptor synthesis and degradation by the density-shift technique.
Highly Cited
1985
Highly Cited
1985
Steroid product-induced, oxygen-mediated damage of microsomal cytochrome P-450 enzymes in Leydig cell cultures. Relationship to desensitization.
Highly Cited
1985
Highly Cited
1985
Interaction of androgens and estrogens in the control of sexual behavior in male Japanese quail
Highly Cited
1981
Highly Cited
1981
Androgens and the thymus.
Tritiated dihydrotestosterone ([3H]DHT) binds with high affinity to a single class of limited capacity sites in cytoplasmic… 
Highly Cited
1980
Highly Cited
1980
Characterization and quantification of the androgen and glucocorticoid receptors in cytosol from rat skeletal muscle.
The binding of the radioactive synthetic hormonal steroids [3H]dexamethasone (9 alpha-fluoro-11 beta, 17 alpha, 21-trihydroxy-16… 
Highly Cited
1978
Highly Cited
1978
Correlation between clinical response to hormone therapy and steroid receptor content in prostatic cancer.
Hormonal therapy is the dominating form of treatment for prostatic carcinoma. The majority of cases (80%) are well controlled for… 
Highly Cited
1976
Highly Cited
1976
Binding of [3H] methyltrienolone (R 1881) in rat prostate and human benign prostatic hypertrophy (BPH)
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