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GR 159897

Known as: GR-159897, GR159897 
National Institutes of Health

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2 relations

Broader (2)

IndolesPiperidines

Papers overview

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2019
2019
Prokinetic effects of the neurokinin NK2 receptor agonist [Lys5,MeLeu9,Nle10]-NKA(4–10) on bladder and colorectal activity in minipigs
2017
2017
NK2 and NK1 receptor-mediated effects of NKA and analogs on colon, bladder, and arterial pressure in anesthetized dogs
Tachykinin NK2 receptor (NK2R) agonists have potential to alleviate clinical conditions associated with bladder and… 
2016
2016
Pharmacodynamic evaluation of Lys5, MeLeu9, Nle10-NKA(4–10) prokinetic effects on bladder and colon activity in acute spinal cord transected and spinally intact rats
The purpose of this study was to determine feasibility of a novel therapeutic approach to drug-induced voiding after spinal cord… 
2012
2012
Non-adrenergic, non-cholinergic, non-purinergic contractions of the urothelium/lamina propria of the pig bladder.
Acetylcholine, and to a lesser extent ATP, mediates neurogenic contractions of bladder smooth muscle. Recently, the urothelium… 
2012
2012
Role of tachykinin and neurokinin receptors in the regulation of ovine omasal contractions
2002
2002
A pharmacophore model for NK2 antagonist comprising compounds from several structurally diverse classes
A neurokinin 2 (NK2) antagonist pharmacophore model has been developed on the basis of five non-peptide antagonists from several… 
2002
2002
Effect of YM-44781, YM-44778 and YM-49598, Novel Tachykinin Antagonists, in a Drug-Induced Bladder Contraction Model
The radioligand binding profiles and in vivo pharmacological characteristics of YM-44781, YM-44778 and YM-49598, novel non… 
1995
1995
Endogenous modulation of excitatory amino acid responsiveness by tachykinin NK1 and NK2 receptors in the rat spinal cord
1 The effects of selective tachykinin (neurokinin, NK) NK1 and NK2 receptor antagonists have been examined on spinal neurones in… 
1995
1995
Analogues of GR159897 a highly potent, non-peptide neurokinin-A NK2 receptor antagonist
1993
1993
GR159897; a potent and selective non-peptide NK2 antagonist
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