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BMS-378806

National Institutes of Health

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Piperazines

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2017
2017
P-D3 Crystal structures of small-molecules HIV-1 entry ihibitor, BMS-378806 and BMS-626529, bound to BG505 SOSIP.664 HIV-1 Env trimer reveal an allosteric competitive etry inhibition mechanism
2013
2013
Is the conformational flexibility of piperazine derivatives important to inhibit HIV-1 replication?
2013
2013
The investigations on HIV-1 gp120 bound with BMS-488043 by using docking and molecular dynamics simulations
BMS-488043, like its predecessor BMS-378806, is a small molecule that can block the interactions between gp120 and CD4, and has… 
2013
2013
Chemically Programmed Antibodies AS HIV-1 Attachment Inhibitors.
Herein we describe the design and application of two small-molecule anti-HIV compounds for the creation of chemically programmed… 
2007
2007
Quantitative determination of BMS-378806 in human plasma and urine by high-performance liquid chromatography/tandem mass spectrometry.
BMS-378806 is a human immunodeficiency virus (HIV) entry inhibitor that is being developed for the oral treatment of HIV… 
2004
2004
Predicted genotypic resistance to the novel entry inhibitor, BMS-378806, among HIV-1 isolates of subtypes A to G
BMS-378806 targets virus entry by inhibiting the binding of HIV-1 gp120 to the CD4 receptor. Env sequences (n = 1226) of subtypes… 
Review
2004
Review
2004
HIV-1 entry inhibitor entrances.
Review
2004
Review
2004
New advances in HIV entry inhibitors development.
Considerable advances have been made in the last years in the design of derivatives acting as inhibitors of HIV entry and fusion… 
2003
2003
Blocking the docking of HIV-1
There are estimated to be >42 million people worldwide who live with HIV-1 infection. Any novel means of treating infection… 
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