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bitolterol

Known as: Bitolterolum, bitolterol [Chemical/Ingredient] 
A diester sympathomimetic amine with bronchodilator activity. As an ester prodrug, bitolterol is hydrolyzed by esterases to its active metabolite… 
National Institutes of Health

Related topics

Related topics

10 relations

Broader (3)

Adrenergic beta-2 Receptor AgonistsBronchodilator AgentsEthanolamines
Adrenergic beta2-Agonists [MoA]AsthmaBronchial SpasmBronchodilation [PE]

Narrower (2)

S-1540bitolterol mesylate

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Review
2012
Review
2012
Bitolterol
SummarySynopsisBitolterol is a β-adrenoceptor agonist which is hydrolysed to colterol by tissue esterases present at high… 
2004
2004
Evaluation of the Utilization Patterns of Leukotriene Modifiers in a Large Managed Care Health Plan
OBJECTIVES: To assess the utilization of leukotriene modifiers (LM) relative to national guidelines and to investigate possible… 
Highly Cited
1989
Highly Cited
1989
Nocturnal asthma therapy. Inhaled bitolterol versus sustained-release theophylline.
Many asthmatics complain of increased symptoms, awakenings, and need for additional medications during the sleeping hours… 
1986
1986
Oral beta 2-selective adrenergic bronchodilators.
Oral beta 2-agonists (carbuterol, pirbuterol, procaterol, bitolterol, clenbuterol) are drugs widely used as bronchodilators. The… 
1984
1984
Bitolterol compared to isoproterenol in advanced chronic obstructive pulmonary disease.
Twenty-eight patients with advanced emphysema and/or chronic bronchitis and severe airflow obstruction were randomly assigned to… 
1981
1981
Enhancement of cardiotoxic effects of beta-adrenergic bronchodilators by aminophylline in experimental animals.
1980
1980
Comparative heart rate effects of oral administration of bitolterol, terbutaline and trimetoquinol in unanesthetized dogs.
Effect of a clinical dose of bitolterol, a new oral bronchodilator via adrenergic beta-receptor, on heart rate was compared with… 
1979
1979
Microencapsulation of bitolterol for controlled release and its effect on bronchodilator and heart rate activities in dogs.
Spheronized cores produced by extrusion and marumerization were microencapsulated with ethylcellulose by organic phase separation… 
1979
1979
The influences of the route of administration on the metabolism and excretion of bitolterol, a new bronchodilator, in the rat.
1. [3H]Bitolterol, an ester prodrug to colterol (N-t-butyl-arterenol), when administered orally, was excreted mostly in the urine… 
1976
1976
Esters of N-tert-butylarterenol. Long-acting new bronchodilators with reduced cardiac effects.
The preparation of various esters of N-tert-butylarterenol is described. Esterification of the phenolic OH groups has increased… 
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