VUF 5455

Known as: 4-methoxy-N-(7-methyl-3-(2-pyridinyl)-1-isoquinolinyl)benzamide, VUF-5455, VUF5455 
 
National Institutes of Health

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3 relations

Broader (3)

BenzamidesIndolesPurinergic P1 Receptor Agonists

Papers overview

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2017
2017
Corriden, Ross and Kilpatrick, Laura E. and Kellam, Barrie and Briddon, Stephen J. and Hill, Stephen J. (2014) Kinetic analysis of antagonist-occupied adenosine-A3 receptors within membrane…
In our previous work, using a fluorescent adenosine-A3 receptor (A3AR) agonist and fluorescence correlation spectroscopy (FCS… (More)
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2014
2014
Kinetic analysis of antagonist-occupied adenosine-A3 receptors within membrane microdomains of individual cells provides evidence of receptor dimerization and allosterism
In our previous work, using a fluorescent adenosine-A3 receptor (A3AR) agonist and fluorescence correlation spectroscopy (FCS… (More)
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2010
2010
The effect of allosteric modulators on the kinetics of agonist-G protein-coupled receptor interactions in single living cells.
Allosteric binding sites on adenosine -A(1) and -A(3) receptors represent attractive therapeutic targets for amplifying, in a… (More)
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Review
2005
Review
2005
Allosteric modulation of the adenosine family of receptors.
Allosteric modulators for adenosine receptors (ARs) are of an increasing interest and may have potential therapeutic advantage… (More)
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2003
2003
Identification of essential residues involved in the allosteric modulation of the human A(3) adenosine receptor.
We examined the effects on allosteric modulation and ligand binding of the mutation of amino acid residues of the human A(3… (More)
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2001
2001
Allosteric modulation of A(3) adenosine receptors by a series of 3-(2-pyridinyl)isoquinoline derivatives.
Allosteric modulators of A(1) and A(2A) adenosine receptors have been described; however, for the A(3) adenosine receptor… (More)
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