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Serotonin 5-HT2 Receptor Antagonists

Known as: Antagonist, 5-HT2, Serotonin 5 HT2 Receptor Antagonists, 5-HT2 Antagonist 
Drugs that bind to but do not activate SEROTONIN 5-HT2 RECEPTORS, thereby blocking the actions of SEROTONIN or SEROTONIN 5-HT2 RECEPTOR AGONISTS… 
National Institutes of Health

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APD791AR 246686Lurasidone HydrochlorideSerotonin 5-HT2A Receptor Antagonists
In Bloodaspects of radiation effectschemical synthesisstandards characteristics

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2004
2004
Nialamide-induced hypermotility in mice treated with inhibitors of monoamine uptake, 5-HT antagonists and lithium
When administered orally to mice 1 h before nialamide 100 mg/kg SC two non-selective and nine selective 5-HT uptake inhibitors… 
1997
1997
New dopaminergic and non-dopaminergic theories in schizophrenia and their therapeutic impact
The dopamine (DA) hypothesis of schizophrenia, postulating that schizophrenia is characterized by increased dopamine function… 
1991
1991
The Effect of Different Serotonergic Drugs in the Learned Helplessness Model of Depression
The effect of subchronic treatment with serotonin agonists and antagonists was tested on rats in an animal model of endogenous… 
1990
1990
Naftidrofuryl Inhibits Contractions to Serotonin in Intact and De‐endothelialized Cerebral Arteries in vitro
Excised segments of rabbit middle cerebral artery were cannulated and perfused in vitro at constant flow (1 ml/min). In vessels… 
Review
1990
Review
1990
Reduction of a distinct pool of monoamines by ketanserin in peripheral tissues
Ketanserin is a prototype of a 5-HT2 antagonist which also has moderate α1-adrenoceptor blocking properties. These properties are… 
1990
1990
Effects of the optical isomers of a novel 5-HT2 antagonist and (-)-Bay K 8644 on spontaneous mechanical activity in rat portal veins.
: The effect of the (+)-enantiomer (Ir) and the (-)-enantiomer (Lu) of a novel 5-HT2 antagonist was studied on spontaneous… 
1988
1988
Local hemodynamic effects of serotonin and ketanserin in healthy subjects: studies in the forearm.
The vascular effects of serotonin and the selective 5-HT2 antagonist ketanserin were investigated in the forearm of healthy… 
1985
1985
Cardiovascular and Blood Gas Responses to Ketanserin in Canine Pulmonary Edema Induced by Oleic Acid
This study was performed to determine the cardiovascular and respiratory effects of ketanserin, a specffic 5-HT2 antagonist… 
Highly Cited
1984
Highly Cited
1984
Three distinct subtypes of serotonergic receptors mediate the triphasic blood pressure response to serotonin in rats.
In pentobarbitone- or urethane-anaesthetized normotensive rats the triphasic pressure response to serotonin (5-HT): a short… 
1983
1983
Divergent effects of pirenperone, a 5-HT2 antagonist, on the pressor and tachycardic responses to 5-HT in guinea-pigs.
The effects of pirenperone and cyproheptadine on the pressor and tachycardic responses to 5-hydroxytryptamine (5-HT) and to… 
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