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MEN 16132

Known as: MEN-16132, MEN16132 
National Institutes of Health

Papers overview

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2013
2013
Blockade of nociceptive sensory afferent activity of the rat knee joint by the bradykinin B2 receptor antagonist fasitibant.
2010
2010
Anti‐inflammatory synergy of MEN16132, a kinin B2 receptor antagonist, and dexamethasone in carrageenan‐induced knee joint arthritis in rats
BACKGROUND AND PURPOSE Bradykinin, through its B2 receptor, is involved in inflammatory processes related to arthropathies. In… 
2010
2010
Differences between zofenopril and ramipril, two ACE inhibitors, on cough induced by citric acid in guinea pigs: role of bradykinin and PGE2
Dry and persistent cough is one of the commonest side effects experienced by patients treated with angiotensin-converting enzyme… 
2010
2010
Bradykinin-Induced Lung Inflammation and Bronchoconstriction: Role in Parainfluenze-3 Virus-Induced Inflammation and Airway Hyperreactivity
Inhaled bradykinin causes bronchoconstriction in asthmatic subjects but not nonasthmatics. To date, animal studies with inhaled… 
2009
2009
Novel effects mediated by bradykinin and pharmacological characterization of bradykinin B2 receptor antagonism in human synovial fibroblasts
Background and purpose:  Bradykinin (BK) and B2 receptors have been implicated in the pathophysiology of osteoarthritis (OA), and… 
2009
2009
Effect of Intra-articular 4-(S)-Amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-8-quinolyloxymethyl)phenylsulfonamido]-tetrahydro-2H-4-pyranylcarbonyl} piperazino)-5-oxopentyl](trimethyl)ammonium…
The present study was designed to investigate the role of bradykinin (BK) in the knee joint osteoarthritis induced by intra… 
2009
2009
Pharmacological characterization of the bradykinin B2 receptor antagonist MEN16132 in rat in vitro bioassays.
2007
2007
Comparative antagonist pharmacology at the native mouse bradykinin B2 receptor: radioligand binding and smooth muscle contractility studies
The aim was to characterize the recently discovered non‐peptide antagonist MEN16132 at the mouse B2 receptor, relative to other… 
2005
2005
MEN16132, a novel potent and selective nonpeptide antagonist for the human bradykinin B2 receptor. In vitro pharmacology and molecular characterization.
2005
2005
MEN16132, a Novel Potent and Selective Nonpeptide Kinin B2 Receptor Antagonist: In Vivo Activity on Bradykinin-Induced Bronchoconstriction and Nasal Mucosa Microvascular Leakage in Anesthetized…
We have tested the activity of 4-(S)-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-8-quinolyloxymethyl)phenylsulfonamido… 
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