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Histamine H1 Antagonists, Non-Sedating

Known as: antihistamine non sedating, antihistamines second generation, H1 Antihistamines, Non-Sedating 
A class of non-sedating drugs that bind to but do not activate histamine receptors (DRUG INVERSE AGONISM), thereby blocking the actions of histamine… 
National Institutes of Health

Related topics

Related topics

18 relations
Anti-Allergic AgentsIn Bloodaspects of radiation effectschemical synthesis

Broader (1)

Antihistamines

Narrower (12)

AstemizoleCetirizineLoratadineOlopatadine hydrochloride

Papers overview

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Review
2014
Review
2014
Evaluation of discharge medication orders following automatic therapeutic substitution of commonly exchanged drug classes.
OBJECTIVE Automatic therapeutic substitution (ATS) is a mechanism that, upon patient hospitalization, prompts the pharmacist to… 
2013
2013
Rupatadine improves quality of life in mastocytosis: a randomized, double‐blind, placebo‐controlled trial
Mastocytosis is frequently associated with mast cell‐mediated symptoms which require relieving medication. While second… 
Review
2007
Review
2007
Long-term issues in the treatment of sleep disorders.
Insomnia is a disorder characterized by chronic sleep disturbance associated with daytime disability or distress, such as memory… 
2005
2005
Metabolism and excretion of loratadine in male and female mice, rats and monkeys
The metabolism and excretion of loratadine (LOR), a long–acting non–sedating antihistamine, have been evaluated in male and… 
2004
2004
The utility of mixed‐effects covariate analysis in rapid selection of doses in pediatric subjects: A case study with fexofenadine hydrochloride
Fexofenadine hydrochloride is a non‐sedating antihistamine that is used in the treatment of symptoms associated with seasonal… 
1999
1999
In vitro inhibition of human liver drug metabolizing enzymes by second generation antihistamines.
1996
1996
Comparison of mizolastine with loratadine in the treatment of perennial allergic rhinitis.
Mizolastine is a new, non-sedating antihistamine providing satisfactory symptomatic relief in seasonal allergic rhinitis. The… 
Review
1996
Review
1996
Antiallergic properties of antihistamines.
Histamine is a major mediator of the allergic reaction, and histamine H1-receptor antagonists have a long history of clinical… 
1988
1988
Efficacy of an oral antihistamine, astemizole, as compared to a nasal steroid spray in hay fever
The efficacy and side effects of the oral H1‐antihistamine, astemizole, were compared with those of nasal beclomethasone in 158… 
1982
1982
Terfenadine, the first non-sedating antihistamine.
Alpha-[4-(1,1-Dimethylethyl)phenyl]-4-(hydroxydiphenylmethyl)- piperidinebutanol (terfenadine, RMI 9918, Triludan, Teldane, resp… 
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