Skip to search formSkip to main content
You are currently offline. Some features of the site may not work correctly.

Diprenorphine

Known as: 6,14-Ethenomorphinan-7-methanol, 17-(cyclopropylmethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-alpha,alpha-dimethyl-, (5alpha,7alpha)-, Diprenorfin, Diprenorphine [Chemical/Ingredient] 
A narcotic antagonist similar in action to NALOXONE. It is used to remobilize animals after ETORPHINE neuroleptanalgesia and is considered a specific… Expand
National Institutes of Health

Related topics

Related topics

10 relations

Narrower (2)

Diprenorphine HydrochlorideRevivon
In Bloodagonistsanalogs & derivativesantagonists & inhibitors
Expand

Broader (1)

Narcotic Antagonists

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Highly Cited
2005
Highly Cited
2005
Identification of the molecular mechanisms by which the diterpenoid salvinorin A binds to kappa-opioid receptors.
Salvinorin A is a naturally occurring hallucinogenic diterpenoid from the plant Salvia divinorumthat selectively and potently… Expand
  • figure 1
  • figure 2
  • figure 3
  • figure 4
  • table 1
Is this relevant?
Highly Cited
2004
Highly Cited
2004
Central poststroke pain and reduced opioid receptor binding within pain processing circuitries: a [11C]diprenorphine PET study
&NA; Based on concepts that endogenous opioids participate in neural transmission of pain, the present study in central… Expand
Is this relevant?
Highly Cited
1999
Highly Cited
1999
Measurement of Changes in Opioid Receptor Binding in Vivo During Trigeminal Neuralgic Pain Using [11C]Diprenorphine and Positron Emission Tomography
The binding of [11C]diprenorphine to µ, κ, and Δ subsites in cortical and subcortical structures was measured by positron… Expand
Is this relevant?
Highly Cited
1999
Highly Cited
1999
Central pain after pontine infarction is associated with changes in opioid receptor binding: a PET study with 11C-diprenorphine.
Using 18F-fluorodeoxyglucose and 11C-diprenorphine positron emission tomography (PET), we investigated alterations in glucose… Expand
  • figure 1
  • figure 2
  • figure 3
Is this relevant?
Highly Cited
1991
Highly Cited
1991
Compartmental Analysis of Diprenorphine Binding to Opiate Receptors in the Rat in vivo and its Comparison with Equilibrium Data in vitro
The regional binding of the opiate receptor ligand diprenorphine has been examined in rat brain both in vivo and in vitro. The… Expand
  • figure 1
  • figure 2
  • table 1
  • figure 4
  • figure 3
Is this relevant?
Highly Cited
1989
Highly Cited
1989
Dual opioid modulation of the action potential duration of mouse dorsal root ganglion neurons in culture
Multiple modulatory effects of opioids on the duration of the calcium component of the action potential (APD) of dorsal-root… Expand
  • figure 1
  • figure 2
  • table II
  • table IV
  • table V
Is this relevant?
Highly Cited
1981
Highly Cited
1981
An autoradiographic map of (3H) diprenorphine binding in rat brain: Effects of social interaction
(3H)Diprenorphine binding was analyzed autoradiographically in the brains of 33 day old rat pups. A photographic atlas of… Expand
Is this relevant?
Highly Cited
1980
Highly Cited
1980
Radioautography of binding of tritiated diprenorphine to opiate receptors in the rat.
Abstract Radioautography of tritiated diprenorphine in rat brain indicates anatomic distribution of receptors with a greater… Expand
Is this relevant?
Highly Cited
1978
Highly Cited
1978
Naloxone as a GABA antagonist: evidence from iontophoretic, receptor binding and convulsant studies.
From the following three lines of evidence, it is proposed that at least part of the convulsant activity of naloxone is a result… Expand
Is this relevant?
Highly Cited
1977
Highly Cited
1977
AGONIST AND ANTAGONIST PROPERTIES OF BUPRENORPHINE, A NEW ANTINOCICEPTIVE AGENT
1 Buprenorphine is a highly lipophilic derivative of oripavine. In rodent antinociceptive assays (writhing, tail pressure… Expand
Is this relevant?
By clicking accept or continuing to use the site, you agree to the terms outlined in our Privacy Policy, Terms of Service, and Dataset License
ACCEPT & CONTINUE