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Celiprolol

Known as: Urea, N'-(3-acetyl-4-(3-((1,1-dimethylethyl)amino)-2-hydroxypropoxy)phenyl)-N,N-diethyl-, RS)-N'-{3-acetyl-4-[3-(tert-butylamino)-2-hydroxypropoxy]phenyl}-N,N-diethylurea, Celiprolol [Chemical/Ingredient] 
A cardioselective beta-1 adrenergic antagonist that has intrinsic symopathomimetic activity. It is used in the management of ANGINA PECTORIS and… 
National Institutes of Health

Related topics

Related topics

16 relations

Broader (5)

Adrenergic beta-1 Receptor AntagonistsAnti-Arrhythmia AgentsAntihypertensive AgentsSympathomimetics
Celiprolol 200 MGIn Bloodagonistsanalogs & derivatives

Narrower (3)

Celiprolol HydrochlorideST-1396Selectol

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2017
2017
Small-Dosing Clinical Study: Pharmacokinetic, Pharmacogenomic (SLCO2B1 and ABCG2), and Interaction (Atorvastatin and Grapefruit Juice) Profiles of 5 Probes for OATP2B1 and BCRP.
Highly Cited
2014
Highly Cited
2014
Single-walled carbon nanotube-based polymer monoliths for the enantioselective nano-liquid chromatographic separation of racemic pharmaceuticals.
Highly Cited
2008
Highly Cited
2008
Effects of the antioxidative beta-blocker celiprolol on endothelial progenitor cells in hypertensive rats.
BACKGROUND Endothelial progenitor cells (EPCs) derived from bone marrow migrate to areas of endothelial damage and repair them… 
Highly Cited
2001
Highly Cited
2001
Quantitative structure-retention and retention-activity relationships of beta-blocking agents by micellar liquid chromatography.
Highly Cited
2001
Highly Cited
2001
A comprehensive account on the role of efflux transporters in the gastrointestinal absorption of 13 commonly used substrate drugs in humans.
BACKGROUND The potential absorption-limiting effect of intestinal efflux transporters such as P-glycoprotein (P-gp) has been well… 
Highly Cited
2000
Highly Cited
2000
A comparative in vitro study of percutaneous penetration of beta-blockers in human skin.
1999
1999
Experimental design for enantioselective separation of celiprolol by capillary electrophoresis using sulfated β‐cyclodextrin
A capillary zone electrophoresis method was developed for the enantioseparation of celiprolol enantiomers, using a sulfated… 
Review
1991
Review
1991
Metabolic considerations in the choice of therapy for the patient with hypertension.
1988
1988
Placental transfer of beta-adrenergic antagonists studied in an in vitro perfusion system of human placental tissue.
Highly Cited
1986
Highly Cited
1986
Celiprolol, atenolol and propranolol: a comparison of pulmonary effects in asthmatic patients.
Celiprolol, a new beta-adrenoceptor antagonist, blocks serotonin- and methacholine-mediated bronchoconstriction in animals, even… 
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