Celiprolol

Known as: Urea, N'-(3-acetyl-4-(3-((1,1-dimethylethyl)amino)-2-hydroxypropoxy)phenyl)-N,N-diethyl-, RS)-N'-{3-acetyl-4-[3-(tert-butylamino)-2-hydroxypropoxy]phenyl}-N,N-diethylurea, Celiprolol [Chemical/Ingredient] 
A cardioselective beta-1 adrenergic antagonist that has intrinsic symopathomimetic activity. It is used in the management of ANGINA PECTORIS and… (More)
National Institutes of Health

Papers overview

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2012
2012
The authors evaluated the contribution of the SLCO2B1 polymorphism to the pharmacokinetics of celiprolol at a microdose (MD) and… (More)
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2009
2009
Gastrointestinal absorption of several beta-blockers is inhibited by citrus juices, although molecular mechanism(s) lying on… (More)
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Highly Cited
2004
Highly Cited
2004
The efflux transporter, P-glycoprotein (P-gp), located in the apical membranes of intestinal absorptive cells, can reduce the… (More)
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2003
2003
Vascular cell adhesion molecule-1 (VCAM-1) and reactive oxygen species play critical roles in early atherogenesis, and nitric… (More)
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2000
Highly Cited
2000
BACKGROUND Local pulse pressure (PP) is an independent determinant of carotid artery wall thickness, stronger than mean blood… (More)
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1994
1994
A decrease in endothelium-derived relaxing factor or nitric oxide has been proposed as a potential mechanism of increased… (More)
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1993
1993
1. The transepithelial transport of the beta-adrenoceptor blocking drug, celiprolol, was investigated in monolayers of the well… (More)
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Highly Cited
1992
Highly Cited
1992
The antioxidant effect of carvedilol, a new vasodilating, beta adrenoceptor blocker was studied and compared with five other beta… (More)
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1991
1991
The comparative antianginal effects and safety of propranolol and celiprolol, a highly beta 1-selective adrenoceptor blocker with… (More)
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1986
1986
Celiprolol, a new beta-adrenoceptor antagonist, blocks serotonin- and methacholine-mediated bronchoconstriction in animals, even… (More)
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