Bupranolol

Known as: 2-Propanol, 1-(2-chloro-5-methylphenoxy)-3-((1,1-dimethylethyl)amino)-, hydrochloride, (+-)-, Bupranol, Bupranolol [Chemical/Ingredient] 
An adrenergic-beta-2 antagonist that has been used for cardiac arrhythmia, angina pectoris, hypertension, glaucoma, and as an antithrombotic.
National Institutes of Health

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Highly Cited
2005
Highly Cited
2005
BACKGROUND The therapeutic effects of nonspecific beta-blockers are limited by vasoconstriction, thus justifying the interest in… (More)
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2005
2005
Bupranolol (BPL) is a suitable drug candidate for transdermal drug delivery system development based on its favorable… (More)
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2004
2004
This study investigates the effect of the aryloxypropanolamines 4-[3-[(1,1-dimethylethyl)amino]-2-hydroxypropoxy]-1,3-dihydro-2H… (More)
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Highly Cited
1999
Highly Cited
1999
PURPOSE To investigate the presence of the beta3-adrenoceptor (beta3-AR) in human and rat detrusor muscle and the usefulness of… (More)
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Highly Cited
1996
Highly Cited
1996
Beta3-adrenoceptors are involved in metabolism, gut relaxation, and vascular vasodilation. However, their existence and role in… (More)
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1992
1992
Transdermal absorption of drugs is limited by the stratum corneum, which serves as a diffusion barrier. This barrier might be… (More)
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1991
1991
Transdermal administration of drugs possesses several advantages in therapy, but is limited by generally poor penetration through… (More)
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1981
1981
A technique is described for the synthesis of 3H-(−)-bupranolol (3H-BU) by tritium exchange. The binding of this new radioligand… (More)
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1980
1980
Melting points measured with the capillary method were 150.5°C, 150.5°C and 224.0°C for hydrochlorides of (+)-bupranolol… (More)
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1980
1980
Localization of instilled 14C-bupranolol was studied in the rabbit eye by means of light microscopic radioautography. After the… (More)
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