Bradykinin Receptor Antagonists

Known as: Receptor Blockers, Bradykinin, Bradykinin Antagonists, Antagonists, Bradykinin Receptor 
Compounds and drugs that inhibit ligand binding or cellular signaling by BRADYKININ RECEPTORS.
National Institutes of Health

Papers overview

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Highly Cited
2002
Highly Cited
2002
M(1) muscarinic (M(1)AChRs) and B(2) bradykinin (B(2)Rs) receptors are two PLCbeta-coupled receptors that mobilize Ca(2+) in… (More)
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2001
2001
Bradykinin has been linked to the development of restenosis in response to vascular injury. We therefore examined the effect of… (More)
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2001
2001
Objective and Design: We studied the ability of bradykinin (BK) receptor antagonists type 1 and 2 (B1-RA, B2-RA) to prevent acute… (More)
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Highly Cited
1998
Highly Cited
1998
The mechanism of the enhanced vascular permeability and retention (EPR) effect seen in solid tumors was investigated with sarcoma… (More)
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1997
1997
We describe the receptor binding and antagonistic properties of two novel nonpeptide antagonists, FR167344 (3-bromo-8-[2,6… (More)
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1997
1997
Bradykinin and lys-bradykinin generated intrarenally appear to be important renal paracrine hormones. However, the renal effects… (More)
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1997
1997
The major isoform of Trypanosoma cruzi cysteinyl proteinase (cruzipain) has generated Lys-bradykinin (Lys-BK or kallidin), a… (More)
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Review
1990
Review
1990
Bradykinin and its active metabolites are produced at the sites of their actions by kallikreins. They potently elicit a variety… (More)
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Highly Cited
1988
Highly Cited
1988
Autoradiographic studies localize [3H]bradykinin receptor binding sites to the substantia gelatinosa, dorsal root, and a subset… (More)
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1988
1988
Glandular kallikreins are a family of proteases encoded by a variable number of genes in different mammalian species. In all… (More)
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