Androgen Receptor Antagonists [MoA]

Known as: Androgen Receptor Antagonists, Androgen Receptor Inhibitor 
 
National Institutes of Health

Topic mentions per year

Topic mentions per year

1998-2016
024619982016

Papers overview

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2012
2012
Previously available androgen receptor (AR) antagonists (bicalutamide, flutamide, and nilutamide) have limited activity against… (More)
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2012
2012
A series of 4-phenylpyrrole derivatives D were designed, synthesized, and evaluated for their potential as novel orally available… (More)
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2012
2012
Androgen receptor antagonists have been proved to be effective anti-prostate cancer agents. 3D-QSAR and Molecular docking methods… (More)
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2011
2011
The studies presented in this manuscript focus on characterization of transcriptomic responses to anti-androgens in zebrafish… (More)
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2011
2011
An aryloxy tetramethylcyclobutane was identified as a novel template for androgen receptor (AR) antagonists via cell-based high… (More)
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2009
2009
Androgen receptor (AR) continues to play a central role in prostate cancers that relapse after androgen deprivation therapy, but… (More)
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2007
2007
The synthesis and in vivo SAR of N-benzyl, N-aceto, and N-ethylene ether derivatives of 2-(2,2,2-trifluoroethyl)-5,6-dichloro… (More)
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2005
2005
A novel series of isoindoledione based compounds were identified as potent antagonists of the androgen receptor (AR). Co… (More)
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2002
2002
A number of curcumin analogues were prepared and evaluated as potential androgen receptor antagonists against two human prostate… (More)
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