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azaphenylalanine

 
National Institutes of Health

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Broader (1)

Phenylalanine
analogs & derivatives

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2013
2013
Benzotriazole-mediated synthesis of aza-peptides: en route to an aza-leuenkephalin analogue.
Novel N-(N-Pg-azadipeptidoyl)benzotriazoles 20a-e couple efficiently with α-amino acids 21a-e, dipeptides 22a-c, aminoxyacetic… Expand
2009
2009
Azaphenylalanine-based serine protease inhibitors induce caspase-mediated apoptosis.
Molecules regulating cell death constitute prominent therapeutic targets. The pro-apoptotic role of serine protease inhibitors… Expand
2007
2007
The beta-turn scaffold of tripeptide containing an azaphenylalanine residue.
The conformational preferences of azaphenylalanine-containing peptide were investigated using a model compound, Ac-azaPhe-NHMe… Expand
2005
2005
Antithrombotic potential of new direct thrombin inhibitors built on the azaphenylalanine scaffold in two rat venous thrombosis models.
The antithrombotic potential of new direct thrombin inhibitors built on the azaphenylalanine scaffold (LK-732, LK-639 and LK-731… Expand
2004
2004
Thrombin inhibitors built on an azaphenylalanine scaffold.
A series of azaphenylalanine derivatives were investigated as novel thrombin inhibitors based on the prodrug principle. By… Expand
2004
2004
Synthesis and in vitro evaluation of new azaphenylalanine derivatives as serine protease inhibitors.
New inhibitors of serine proteases with azaphenylalanine scaffold were synthesized and their activity was evaluated in vitro. We… Expand
2004
2004
Novel non-covalent azaphenylalanine thrombin inhibitors with an aminomethyl or amino group at the P1 position.
Design, synthesis and biological evaluation of a series of novel non-covalent azaphenylalanine thrombin inhibitors are presented… Expand
2001
2001
Design and structure-activity relationship of thrombin inhibitors with an azaphenylalanine scaffold: potency and selectivity enhancements via P2 optimization.
Theoretical and structural studies followed by the directed synthesis and in vitro biological tests lead us to novel noncovalent… Expand
2001
2001
Novel thrombin inhibitors with azaphenylalanine scaffold.
In this paper the synthesis and antithrombotic activity of a series of novel thrombin inhibitors with azaphenylalanine scaffold… Expand
1978
1978
Synthesis and biological activity of highly active alpha-aza analogues of luliberin.
Analogues of luliberin containing an alpha-azaamino acid in position 6, 9, or 10 (I--XIV) have been synthesized by the solution… Expand
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