azaphenylalanine

 
National Institutes of Health

Topic mentions per year

Topic mentions per year

1978-2012
012319782012

Papers overview

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2012
2012
Serine proteases have proven to be promising pharmacological targets in contemporary drug discovery for cancer treatment. Since… (More)
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2009
2009
Molecules regulating cell death constitute prominent therapeutic targets. The pro-apoptotic role of serine protease inhibitors… (More)
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2007
2007
The conformational preferences of azaphenylalanine-containing peptide were investigated using a model compound, Ac-azaPhe-NHMe… (More)
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2007
2007
Design, synthesis and biochemical evaluation of a series of novel non-covalent thrombin inhibitors with a 1-amidinopiperidine… (More)
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2006
2006
The main structural feature of direct thrombin inhibitor LK-732 responsible for the appropriate interaction at the thrombin… (More)
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2005
2005
The antithrombotic potential of new direct thrombin inhibitors built on the azaphenylalanine scaffold (LK-732, LK-639 and LK-731… (More)
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2004
2004
A series of azaphenylalanine derivatives were investigated as novel thrombin inhibitors based on the prodrug principle. By… (More)
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2004
2004
Design, synthesis and biological evaluation of a series of novel non-covalent azaphenylalanine thrombin inhibitors are presented… (More)
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2004
2004
New inhibitors of serine proteases with azaphenylalanine scaffold were synthesized and their activity was evaluated in vitro. We… (More)
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2001
2001
In this paper the synthesis and antithrombotic activity of a series of novel thrombin inhibitors with azaphenylalanine scaffold… (More)
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