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artemisone

Known as: 4-((3R,5AS,6R,8aS,9R,10R,12R,12aR)-3,6,9-Trimethyldecahydro-12H-3,12-Epoxypyrano(4,3-J)(1,2)Benzodioxepin-10-yl)Thiomorpholine-1,1-Dione, Artemifone 
National Institutes of Health

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Related topics

1 relation

Broader (1)

Artemisinins

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2020
2020
Optimal 10-Aminoartemisinins With Potent Transmission-Blocking Capabilities for New Artemisinin Combination Therapies–Activities Against Blood Stage P. falciparum Including PfKI3 C580Y Mutants and…
We have demonstrated previously that amino-artemisinins including artemiside and artemisone in which an amino group replaces the… 
2018
2018
Formulation of Natural Oil Nano-Emulsions for the Topical Delivery of Clofazimine, Artemisone and Decoquinate
The aim of this study was to formulate nano-emulsions comprising natural oils and the active pharmaceutical ingredients (APIs… 
2016
2016
Methylene Homologues of Artemisone: An Unexpected Structure–Activity Relationship and a Possible Implication for the Design of C10‐Substituted Artemisinins
We sought to establish if methylene homologues of artemisone are biologically more active and more stable than artemisone. The… 
2016
2016
In vitro activity of artemisone and artemisinin derivatives against extracellular and intracellular Helicobacter pylori.
2014
2014
Ex Vivo Activity of Endoperoxide Antimalarials, Including Artemisone and Arterolane, against Multidrug-Resistant Plasmodium falciparum Isolates from Cambodia
ABSTRACT Novel synthetic endoperoxides are being evaluated as new components of artemisinin combination therapies (ACTs) to treat… 
2014
2014
Inhibition of metalloproteinase-9 secretion and gene expression by artemisinin derivatives.
2014
2014
Treatment of Murine Cerebral Malaria by Artemisone in Combination with Conventional Antimalarial Drugs: Antiplasmodial Effects and Immune Responses
ABSTRACT The decreasing effectiveness of antimalarial therapy due to drug resistance necessitates constant efforts to develop new… 
2011
2011
Second-Generation Peroxides: The OZs and Artemisone
The emergence of multi-drug resistant strains of Plasmodium falciparum has rendered many affordable antimalarials, such as… 
2010
2010
Artemisone Uptake in Plasmodium falciparum-Infected Erythrocytes
ABSTRACT Artemisone is one of the most promising artemisinin derivatives in clinical trials. Previous studies with radiolabeled… 
2006
2006
In vitro activity of artemisone compared with artesunate against Plasmodium falciparum.
Artemisinins show the potential for neurotoxicity in preclinical studies. Artemisone is a leading candidate of second-generation… 
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