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antarelix

Known as: D-Alaninamide, N-acetyl-3-(2-naphthalenyl)-D-alanyl-4-chloro-D-phenylalanyl-3-(3-pyridinyl)-D-alanyl-L-seryl-L-tyrosyl-N6-(aminocarbonyl)-D-lysyl-L-leucyl-N6-(1-methylethyl)-L-lysyl-L-prolyl-, teverelix acetate, teverelix 
 
National Institutes of Health

Related topics

Related topics

3 relations

Narrower (1)

EP 24332

Broader (2)

Hormone AntagonistsOligopeptides

Papers overview

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Highly Cited
2012
Highly Cited
2012
RF9 Powerfully Stimulates Gonadotrophin Secretion in the Ewe: Evidence for a Seasonal Threshold of Sensitivity
GPR147 and its endogenous ligands, RFRPs, are emerging as important actors in hypothalamic‐pituitary axis control. The role of… Expand
2004
2004
Effect of p-chlorophenylalanine on the loss and maintenance of tolerance to ethanol
Rats were rendered tolerant to the motor-impairing effects of ethanol by daily oral administration. Subsequently, ethanol was… Expand
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2004
2004
Effect of GnRH antagonists treatment on gonadotrophin secretion, follicular development and inhibin A secretion in goats.
The aim of this study was to determine, for goats, the effects of daily doses of GnRH antagonist on ovarian endocrine and… Expand
2003
2003
PLGA-PEG microspheres of teverelix: influence of polymer type on microsphere characteristics and on teverelix in vitro release.
Teverelix microspheres were produced by coacervation using a new type of poly(ester-carbonates) made of block copolymers of poly… Expand
2003
2003
Use of a GnRH antagonist, antarelix, associated or not with hCG, to control ovulation in cyclic pony mares.
The GnRH antagonist antarelix (Teverelix) was administered to mares (0.01 mg/kg, i.v., twice a day) during the periovulatory… Expand
Highly Cited
2002
Highly Cited
2002
Sequential role of e2 and GnRH for the expression of estrous behavior in ewes.
Preovulatory GnRH secretion in ewes, measured in portal blood and cerebrospinal fluid, starts at the time of the LH surge… Expand
2000
2000
Pituitary and gonadal endocrine effects and pharmacokinetics of the novel luteinizing hormone‐releasing hormone antagonist teverelix in healthy men—a first‐dose‐in‐humans study
Teverelix is a novel synthetic peptidic luteinizing hormone‐releasing hormone (LHRH) antagonist. 
1993
1993
Antarelix (EP 24332) a novel water soluble LHRH antagonist.
A novel water soluble LHRH antagonist (EP 24332-Antarelix) is described. Its activity in vitro and in vivo in several animal… Expand
1987
1987
Enantiomeric composition analysis of amphetamine and methamphetamine by chiral phase high-performance liquid chromatography-mass spectrometry.
N-(Trifluoroacetyl)-l-prolyl- (N-TFA-l-prolyl-) d- and l-amphetamine diastereoisomers were separated by high-performance liquid… Expand
1986
1986
Effects of 15(R)-15-methyl prostaglandin E2 (arbaprostil) on gastric secretion and various gastric lesions induced in rats.
We studied the effects of 15(R)-15-methyl prostaglandin E2 (arbaprostil) on gastric secretion and various acute and chronic… Expand
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