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Thiazepines

Known as: Thiazepines [Chemical/Ingredient], thiazepine 
National Institutes of Health

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1,5-benzothiazepine2164U902169W 94264W 94
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Papers overview

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Highly Cited
2011
Highly Cited
2011
Coumarin‐Based Bioactive Compounds: Facile Synthesis and Biological Evaluation of Coumarin‐Fused 1,4‐Thiazepines
As part of our ongoing studies on the synthesis of bioactive coumarin compounds, we synthesized a series of new coumarin‐fused 1… 
2008
2008
Concise assembly of highly substituted furan-fused 1,4-thiazepines and their Diels-Alder reactions with benzynes.
A facile and highly efficient three-component reaction of thiazole or benzothiazole carbenes, disubstituted ketenes, and… 
2006
2006
Structure-activity relationship of 6-methylidene penems bearing 6,5 bicyclic heterocycles as broad-spectrum beta-lactamase inhibitors: evidence for 1,4-thiazepine intermediates with C7 R…
The design and synthesis of a series of 6-methylidene penems containing [6,5]-fused bicycles (thiophene, imidazole, or pyrazle… 
Highly Cited
2004
Highly Cited
2004
Structure-activity relationship of 6-methylidene penems bearing tricyclic heterocycles as broad-spectrum beta-lactamase inhibitors: crystallographic structures show unexpected binding of 1,4…
The design and synthesis of a series of seven tricyclic 6-methylidene penems as novel class A and C serine beta-lactamase… 
2004
2004
Synthesis of novel thiazolothiazepine based HIV-1 integrase inhibitors.
2003
2003
An efficient assembly of heterobenzazepine ring systems utilizing an intramolecular palladium-catalyzed cycloamination.
Azaheterocyclic compounds are interesting and medicinally relevant targets. Herein we disclose an improved synthesis into the… 
Highly Cited
1999
Highly Cited
1999
Design, synthesis, and biological evaluation of potent thiazine- and thiazepine-based matrix metalloproteinase inhibitors.
The synthesis and enzyme inhibition data for a series of thiazine- and thiazepine-based matrix metalloproteinase (MMP) inhibitors… 
Highly Cited
1997
Highly Cited
1997
Regulation of retinoidal actions by diazepinylbenzoic acids. Retinoid synergists which activate the RXR-RAR heterodimers.
In human HL-60 promyelocytic leukemia cells, diazepinylbenzoic acid derivatives can exhibit either antagonistic or synergistic… 
Highly Cited
1994
Highly Cited
1994
Pyridobenzoxazepine and pyridobenzothiazepine derivatives as potential central nervous system agents: synthesis and neurochemical study.
In order to characterize the pharmacological profile of the different chemical classes of pyridobenzazepine derivatives, a series… 
Highly Cited
1988
Highly Cited
1988
Structural dependency of the inhibitory action of benzodiazepines and related compounds on the mitochondrial Na+-Ca2+ exchanger.
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