Skip to search formSkip to main content
You are currently offline. Some features of the site may not work correctly.

1,5-benzothiazepine

 
National Institutes of Health

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Highly Cited
2015
Highly Cited
2015
The 1,5-benzothiazepine moiety is well-known as a versatile pharmacophore, and its derivatives are expected to have antagonism… Expand
  • figure 1
  • table 1
  • table 2
2009
2009
Two series of novel 1,5-benzothiazepine derivatives (23 compounds) were efficiently synthesized and evaluated for antibacterial… Expand
  • figure 1
  • table 1
  • table 2
  • figure 3
  • figure 2
1991
1991
In an attempt to improve the effectiveness and duration of the action of diltiazem (1), a 1,5-benzothiazepine calcium channel… Expand
1988
1988
Effects of TA-3090 ((+) (2S,3S)-3-acetoxy-8-chloro-5-(2-(dimethylamino)ethyl)-2, 3-dihydro-2-(4-methoxyphenyl)-1,5-benzothiazepin… Expand
1986
1986
A seires of (R)-3-amino-4-oxo-2, 3, 4, 5-tetrahydro-1, 5-benzothiazepine-5-acetic acids (8) and (S)-3-amino-4-oxo-2, 3, 4, 5… Expand
Highly Cited
1985
Highly Cited
1985
The synthesis of chiral 1,5-benzothiazepines 2a-c, 14a-c, 15c, and 16a prepared from cysteine is described. In vitro inhibition… Expand
Highly Cited
1975
Highly Cited
1975
Diltiazem, a new 1,5-benzothiazepine derivative, antagonized calcium ion and thus caused a reduction in the contractile force of… Expand
1974
1974
Abstract Effects of a new coronary vasodilator, CRD-401, on renal blood flow and renal function were investigated in anesthetized… Expand
Highly Cited
1973
Highly Cited
1973
The coronary vasodilating action of 1, 5-benzothiazepine derivatives and the structureactivity relationship were examined in the… Expand
Highly Cited
1972
Highly Cited
1972
Abstract 3-Acetoxy-2, 3-dihydro-5-[2-(dimethylamino)ethyl]-2-(p-methoxyphenyl)-l, 5-benzothia-zepin-4(5H)-one hydrochloride is a… Expand