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Neurokinin-1 Receptor Antagonists
Known as:
Receptor Blockers, Neuroleukin-1
, Receptor Antagonists, Neurokinin-1
, Neurokinin 1 Receptor Antagonists
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Compounds that inhibit or block the activity of NEUROKININ-1 RECEPTORS.
National Institutes of Health
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Related topics
Related topics
29 relations
Narrower (25)
AZD 2738
AZD 8081
CAM 4515
CI 1021
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In Blood
aspects of radiation effects
chemical synthesis
standards characteristics
Papers overview
Semantic Scholar uses AI to extract papers important to this topic.
2010
2010
Use of neurokinin-1 receptor antagonists in patients receiving moderately or highly emetogenic chemotherapy.
M. Rogers
,
L. Blackburn
Clinical Journal of Oncology Nursing
2010
Corpus ID: 26937135
Chemotherapy-induced nausea and vomiting (CINV) is a serious adverse effect of chemotherapy that limits patients' physical…
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2009
2009
Potent, brain-penetrant, hydroisoindoline-based human neurokinin-1 receptor antagonists.
Jinlong Jiang
,
J. Bunda
,
+19 authors
S. Mills
Journal of Medicinal Chemistry
2009
Corpus ID: 29677139
3-[(3aR,4R,5S,7aS)-5-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}-4-(4-fluorophenyl)octahydro-2H-isoindol-2-yl]cyclopent-2-en…
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2009
2009
Synergy between microtubule destabilizing agents and neurokinin 1 receptor antagonists identified by an siRNA synthetic lethal screen
C. Kitchens
,
Peter R McDonald
,
I. Pollack
,
P. Wipf
,
J. Lazo
2009
Corpus ID: 82026016
Coordinated microtubule polymerization and depolymerization is essential for numerous biological functions, including mitotic…
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2007
2007
Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists.
Takashi Yamamoto
,
P. Nair
,
+9 authors
V. Hruby
Journal of Medicinal Chemistry
2007
Corpus ID: 34506085
A series of bifunctional peptides that act as agonists for delta and mu opioid receptors with delta selectivity and as antagonist…
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Review
2004
Review
2004
Potential therapeutic targets for neurokinin-1 receptor antagonists
R. Duffy
2004
Corpus ID: 196359046
The peptide substance P and its tachykinin receptor, neurokinin-1 (NK1), have been the focus of considerable research for their…
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2004
2004
Inhibiting substance p pathway for prevention of chemotherapy-induced emesis: preclinical data, clinical trials of neurokinin-1 receptor antagonists.
R. Navari
Supportive Cancer Therapy
2004
Corpus ID: 23865986
Neurokinin-1 (NK-1) receptor antagonists are a new class of antiemetic agents that have activity in controlling cisplatin-induced…
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Review
2004
Review
2004
Role of Neurokinin-1 Receptor Antagonists in Chemotherapy-Induced Emesis: Summary of Clinical Trials
R. Navari
Cancer Investigation
2004
Corpus ID: 21507821
Chemotherapy-induced nausea and vomiting (CINV) is associated with a significant deterioration in quality of life, and although…
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2001
2001
Neurokinin‐1 Receptor Antagonists Block Acute Cocaine‐Induced Horizontal Locomotion
Madelyne Kraft
,
Sonia Ahluwahlia
,
J. Angulo
Annals of the New York Academy of Sciences
2001
Corpus ID: 27464406
Abstract: Systemic exposure to neurokinin‐1 receptor antagonists CP099994 or LY306740 prior to cocaine administration (10 mg/kg i…
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Highly Cited
1999
Highly Cited
1999
Tachykinin receptors are involved in the “local efferent” motor response to capsaicin in the guinea-pig small intestine and oesophagus
L. Barthó
,
L. Lénárd
,
+4 authors
C. A. Maggi
Neuroscience
1999
Corpus ID: 30469125
1999
1999
Distribution of Fos-like immunoreactivity in guinea-pig brain following administration of the neurokinin-1 receptor agonist, [Sar9,Met(O2)11]substance P
J. Yip
,
L. Chahl
Neuroscience
1999
Corpus ID: 45538734
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