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E 3040

Known as: E-3040, E3040 
 
National Institutes of Health

Related topics

Related topics

3 relations

Broader (2)

BenzothiazolesPyridines

Narrower (1)

E3040 sulfate

Papers overview

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2011
2011
Interactions of urate transporter URAT1 in human kidney with uricosuric drugs.
AIM Hyperuricaemia is a significant factor in a variety of diseases, including gout and cardiovascular diseases. The kidney plays… Expand
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2009
2009
Construction of Triple-Transfected Cells [Organic Anion-Transporting Polypeptide (OATP) 1B1/Multidrug Resistance-Associated Protein (MRP) 2/MRP3 and OATP1B1/MRP2/MRP4] for Analysis of the Sinusoidal…
Multidrug resistance-associated protein (MRP) 3/ABCC3 and MRP4/ABCC4 are ATP-binding cassette (ABC) transporters expressed in the… Expand
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2005
2005
Role of Breast Cancer Resistance Protein (Bcrp1/Abcg2) in the Extrusion of Glucuronide and Sulfate Conjugates from Enterocytes to Intestinal Lumen
The purpose of this study is to examine the significance of efflux transporters in the small intestine to extrude glucuronide (G… Expand
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Highly Cited
2004
Highly Cited
2004
Impaired renal excretion of 6-hydroxy-5,7-dimethyl-2-methylamino-4-(3-pyridylmethyl) benzothiazole (E3040) sulfate in breast cancer resistance protein (BCRP1/ABCG2) knockout mice.
Murine breast cancer resistance protein 1 (Bcrp1) is expressed in the brush-border membrane of proximal tubule cells of the… Expand
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2001
2001
In vitro effects of E3040, a dual inhibitor of 5-lipoxygenase and thromboxane A(2) synthetase, on eicosanoid production.
In vitro pharmacological profiles of E3040, 6-hydroxy-5, 7-dimethyl-2-(methylamino)-4-(3-pyridylmethyl) benzothiazole were… Expand
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2001
2001
Effect of E3040, an inhibitor of 5-lipoxygenase and thromboxane synthase, on rat bowel damage induced by lipopolysaccharide.
Intravenous administration of lipopolysaccharide to rats that had been immunized with lipopolysaccharide induced hemorrhagic… Expand
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Highly Cited
1999
Highly Cited
1999
Characterization of the Transport Properties of Cloned Rat Multidrug Resistance-associated Protein 3 (MRP3)*
We have previously cloned rat MRP3 as an inducible transporter in the liver (Hirohashi, T., Suzuki, H., Ito, K., Ogawa, K., Kume… Expand
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1999
1999
Contribution of organic anion transporting polypeptide to uptake of its possible substrates into rat hepatocytes.
Organic anion transporting polypeptide (oatp1) has been cloned from rat liver as one of the transporters responsible for the… Expand
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1997
1997
Carrier-mediated active transport of the glucuronide and sulfate of 6-hydroxy-5,7-dimethyl-2-methylamino-4-(3-pyridylmethyl) benzothiazole (E3040) into rat liver: quantitative comparison of…
The hepatic uptake of glucuronic acid and sulfate conjugates of 6-hydroxy-5,7-dimethyl-2-methylamino-4-(3-pyridylmethyl… Expand
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1995
1995
Kinetic Analysis of Hepatobiliary Transport for Conjugated Metabolites in the Perfused Liver of Mutant Rats (EHBR) with Hereditary Conjugated Hyperbilirubinemia
AbstractPurpose. Previously, we found that the biliary excretion of the 6-hydroxy-5,7-dimethyl-2-methylamino-4-(3-pyridylmethyl… Expand
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