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Devazepide

Known as: (S)-N-(2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)indole-2-carboxamide, 1H-Indole-2-carboxamide, N-(2,3-dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)-, (S)-, Devazepide [Chemical/Ingredient] 
A derivative of benzodiazepine that acts on the cholecystokinin A (CCKA) receptor to antagonize CCK-8's (SINCALIDE) physiological and behavioral… 
National Institutes of Health

Related topics

Related topics

10 relations

Broader (1)

Hormone Antagonists
In Bloodagonistsanalogs & derivativesantagonists & inhibitors

Narrower (2)

L-364,718MK-329

Papers overview

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2015
2015
Design and synthesis of dialkyoxy-indole-2-carboxamide and dialkyoxy-chromen-2-one as potential CB2 receptor ligands
2014
2014
CP55,940 (−)-cis-3-[2-hydroxy-4-(1,1-dimethylheptyl)phenyl]-trans-4-(3- hydroxypropyl)cyclohexanol GIRK G protein-coupled inwardly-rectifying potassium channel GPCR G protein-coupled receptor GTPγS…
2011
2011
Participación de los receptores de Gastrina / Colecistokinina, y su interacción con la Melatonina en el crecimiento y diferenciación de células HT-29 de cáncer de colon
Tesis Univ. Granada. Departamento de Cirugia y sus Especialidades. Departamento de Fisiologia. Leida en diciembre de 2000 
2007
2007
N-(aminoheteroaryl)-1H-indole-2-carboxamide derivatives as antagonist of TRPV1 or VR1 receptor, preparation thereof and therapeutic use thereof
The present invention relates to formula (I): wherein X1 represents a hydrogen atom or a halogen atom or a C1-C6- alkyl, C3-C7… 
2004
2004
Apolipoprotein AIV stimulates duodenal vagal afferent activity to inhibit gastric motility via a CCK 1 pathway
J. Glatzle, N. Darcel, A. J. Rechs, T. J. Kalogeris, P. Tso, and H. E. Raybould Department of Anatomy, Physiology, and Cell… 
1999
1999
CCK-A receptor antagonists have selective effects on nutrient-induced food intake suppression in rats
Trigazis, L., F. J. Vaccarino, C. E. Greenwood, and G. H. Anderson. CCK-A receptor antagonists have selective effects on nutrient… 
1993
1993
Enterochromaffin-like cells in rat stomach respond to short-term infusion of high doses of cholecystokinin but not to long-term, sustained, moderate hyperCCKemia caused by continuous cholecystokinin…
The histamine-producing enterochromaffin-like (ECL) cells in the oxyntic mucosa are controlled by gastrin. An acute gastrin… 
1993
1993
Characterization of CCK receptors in a novel smooth muscle preparation from the guinea‐pig stomach by use of the selective antagonists CI‐988, L‐365,260 and devazepide
1 The cholecystokinin receptors mediating motor responses in a novel smooth muscle preparation from the corpus region of the… 
1993
1993
Portacaval shunt increases the trophic effect of cholecystokinin on the rat pancreas.
The trophic effect of cholecystokinin (CCK) on the pancreas was examined in portacava-shunted (PCS) rats. Exogenous CCK-8s and… 
1992
1992
Pancreatic atrophy in rats produced by the cholecystokinin-A receptor antagonist devazepide.
According to recent reports, the powerful and selective cholecystokinin (CCK)-A receptor antagonist devazepide (also referred to…