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CH 275

Known as: CH-275 
National Institutes of Health

Related topics

Related topics

2 relations

Broader (1)

Somatostatin
analogs & derivatives

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2012
2012
[Development of non-hormonal regulators of adenylyl cyclase signaling system on the basis of peptides, derivatives of the third intracellular loop of somatostatin receptors].
In the majority of the serpentine type receptors the third intracellular loop (ICL-3) is responsible for interaction with… 
2004
2004
Cellular actions of somatostatin on rat periaqueductal grey neurons in vitro
Functional studies indicate that the midbrain periaqueductal grey (PAG) is involved in the analgesic actions of somatostatin… 
2004
2004
Peptide‐chelating agent conjugate for selective targeting of somatostatin receptor type 1: Synthesis and characterization
Previously reported results suggest that the analogue of the somatostatin des‐AA1,2,5[D‐Trp8,IAmp9]‐somatostatin (CH‐275) peptide… 
Review
2002
Review
2002
Drug design at peptide receptors: somatostatin receptor ligands.
Somatostatin (SRIF, somatotropin release inhibiting factor), discovered for its inhibitory action on growth hormone (GH… 
Highly Cited
2001
Highly Cited
2001
In Vivo Internalization of the Somatostatin sst2A Receptor in Rat Brain: Evidence for Translocation of Cell-Surface Receptors into the Endosomal Recycling Pathway
To determine whether cellular compartmentalization of somatostatin receptors can be regulated in vivo, we examined the… 
Highly Cited
2000
Highly Cited
2000
Somatostatin modulation of excitatory synaptic transmission between periventricular and arcuate hypothalamic nuclei in vitro.
Hypophysiotropic somatostatin (SRIF) and growth hormone-releasing hormone (GHRH) neurons are primarily involved in the… 
2000
2000
Receptor‐mediated internalization of somatostatin in rat cortical and hippocampal neurons
Binding of neuropeptides to their receptors usually results in internalization of receptor‐ligand complexes. This process serves… 
2000
2000
Effects of Somatostatin and Its Analogues on Tyrosine Kinase Activity in Rodent Tumors
The effects of native somatostatin-14 (SS-14) and of its two analogues, octreotide and CH-275, on the activity of tyrosine… 
1998
1998
A somatostatin receptor 1 selective ligand inhibits Ca2+ currents in rat insulinoma 1046‐38 cells
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