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tracazolate

Known as: 4-butylamine-1-ethyl-6-methyl-pyrazolo(3,4)pyridine-5-carboxylic acid ethyl ester 
National Institutes of Health

Related topics

Related topics

2 relations

Narrower (1)

ICI 136,753

Broader (1)

Pyrazoles

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Review
2015
Review
2015
Allosteric modulation of GABAA receptors via multiple drug-binding sites.
  • W. Sieghart
  • Advances in pharmacology
  • 2015
  • Corpus ID: 25109680
Highly Cited
2002
Highly Cited
2002
Tracazolate Reveals a Novel Type of Allosteric Interaction with Recombinant γ-Aminobutyric AcidA Receptors
Tracazolate, a pyrazolopyridine, is an anxiolytic known to interact with gamma-aminobutyric acid (GABA)(A) receptors, adenosine… 
1991
1991
A rapid screening method for the assessment of benzodiazepine receptor-related physical dependence in mice. Evaluation of benzodiazepine-related agonists and partial agonists.
Highly Cited
1988
Highly Cited
1988
Non-xanthine heterocycles: activity as antagonists of A1- and A2-adenosine receptors.
Highly Cited
1986
Highly Cited
1986
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: A novel test of anxiety in the rat
Highly Cited
1986
Highly Cited
1986
Aversive and appetitive properties of anxiogenic and anxiolytic agents
  • S. File
  • Behavioural Brain Research
  • 1986
  • Corpus ID: 4015055
Highly Cited
1983
Highly Cited
1983
Specific high-affinity binding sites for [3H]Ro 5-4864 in rat brain and kidney.
The binding of the novel ligand [3H]Ro 5-4864 to membrane preparations of rat kidney and brain was studied. [3H]Ro 5-4864 binds… 
Review
1983
Review
1983
Novel non-benzodiazepine anxiolytics
Highly Cited
1982
Highly Cited
1982
Differential antagonism of the anticonflict effects of typical and atypical anxiolytics.
Highly Cited
1981
Highly Cited
1981
Perturbation of benzodiazepine receptor binding by pyrazolopyridines involves picrotoxinin/barbiturate receptor sites
The two pyrazolopyridines, etazolate (SQ20009) and cartazolate (SQ65396), enhance the binding of [3H]diazepam to benzodiazepine… 
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