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rolapitant

Known as: 1,7-diazaspiro(4.5)decan-2-one, 8-(((1R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)methyl)-8-phenyl-, (5S,8S)- 
National Institutes of Health

Papers overview

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2018
2018
Purpose: Prevention of chemotherapy-induced nausea and vomiting (CINV) is essential to preserve quality of life in cancer… 
2017
2017
The invention discloses a method for synthesizing a rolapitant intermediate. The method comprises a recrystallization method for… 
2017
2017
The FDA has approved rolapitant injectable emulsion in combination with other antiemetics in adults to prevent delayed… 
Review
2017
Review
2017
Objective: The objective of this selective EBM review is to determine whether or not rolapitant is safe and effective in reducing… 
Review
2017
Review
2017
Neurokinin-1 receptor antagonist, 5-hydroxytryptamine-3 RA, and dexamethasone combination therapy is standard of care for the… 
2017
2017
Rolapitant plus 5-HT3 receptor antagonist and dexamethasone is well tolerated and more effectively controls chemotherapy-induced… 
2016
2016
Rolapitant is a novel NK1 receptor antagonist that maintains >90% receptor binding up to five days after a single 180-mg dose. 
Review
2014
Review
2014
Chemotherapy-induced nausea and vomiting (CINV) has long been one of the most troublesome adverse effects of chemotherapy… 
2014
2014
ABSTRACT Aim: Rolapitant is a highly selective competitive long acting NK-1 receptor antagonist that demonstrated safety and…