clobenpropit

Known as: Carbamimidothioic acid, ((4-chlorophenyl)methyl)-, 3-(1H-imidazol-4-yl)propyl ester, S-(3-(4(5)-imidazolyl))propyl-N-(4-chlorobenzyl)isothiourea 
 
National Institutes of Health

Topic mentions per year

Topic mentions per year

1993-2017
051019932017

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2015
2015
BACKGROUND Histamine is a modulatory neurotransmitter regulating neuronal activity. Antidepressant drugs target modulatory… (More)
  • figure 2
Is this relevant?
2011
2011
UNLABELLED Cholangiocarcinoma (CCA) is a biliary cancer arising from damaged bile ducts. Epithelial-mesenchymal transition (EMT… (More)
  • figure 1
  • figure 2
  • figure 3
  • figure 4
  • figure 5
Is this relevant?
Highly Cited
2004
Highly Cited
2004
1. During mast cell degranulation, histamine is released in large quantities. Human eosinophils were found to express histamine H… (More)
Is this relevant?
2004
2004
This study was performed to investigate whether or not the histamine H3-antagonist clobenpropit can ameliorate spatial memory… (More)
Is this relevant?
Highly Cited
2000
Highly Cited
2000
Recently cDNA encoding the histamine H3 receptor was isolated after 15 years of considerable research. However, several studies… (More)
  • figure 1
  • table I
  • figure 2
  • figure 3
  • figure 4
Is this relevant?
1998
1998
We investigated the effect of the new potent and selective histamine H3 receptor agonist, immepip, and the histamine H3 receptor… (More)
Is this relevant?
Highly Cited
1996
Highly Cited
1996
1. The effects of histamine and agents at histamine receptors on spontaneous and 100 mM K(+)-evoked release of acetylcholine… (More)
Is this relevant?
1994
1994
The effect of clobenpropit (VUF-9153), a new histamine H3 receptor antagonist, on electrically induced convulsions was studied in… (More)
Is this relevant?
1993
1993
We determined the affinities of nordimaprit, homodimaprit, clobenpropit and imetit for H3 binding sites (labelled by 3H-N… (More)
  • figure 1
  • figure 2
  • table 1
  • figure 3
  • figure 4
Is this relevant?
1993
1993
The pharmacological activity of the histamine H3 receptor antagonist VUF 9153 (S-[3-(4(5)-imidazolyl)]propyl-N-(4-chlorobenzyl… (More)
Is this relevant?