aziridine-2,3-dicarboxylate

 
National Institutes of Health

Topic mentions per year

Topic mentions per year

2000-2016
012320002016

Papers overview

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2016
2016
Leishmaniasis is one of the major neglected tropical diseases of the world. Druggable targets are the parasite cysteine proteases… (More)
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2010
2010
The papain-like cysteine cathepsins expressed by Leishmania play a key role in the life cycle of these parasites, turning them… (More)
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2009
2009
Quantum chemical computations on appropriate model systems are used for a rational design of aziridine-based inhibitors of… (More)
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2006
2006
The protozoan parasite Trypanosoma brucei causes Human African trypanosomiasis, which is fatal if left untreated. Due to the… (More)
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2006
2006
To enable a rational design of improved cysteine protease inhibitors, the present work investigates trends in the inhibition… (More)
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2006
2006
A comprehensive screening of N-acylated aziridine (aziridide) based cysteine protease inhibitors containing either Boc-Leu-Caa… (More)
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2004
2004
Cysteine proteases have been implicated in a variety of processes essential for the survival and progression of the malarial… (More)
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2000
2000
Peptides containing aziridine-2,3-dicarboxylate (Azi) as electrophilic building block are evaluated as inhibitors of the cysteine… (More)
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