Skip to search formSkip to main contentSkip to account menu

GSK 189254

Known as: GSK-189254, GSK189254 
National Institutes of Health

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2016
2016
Discovery and Preclinical Validation of [(11)C]AZ13153556, a Novel Probe for the Histamine Type 3 Receptor.
UNLABELLED The histamine type 3 receptor (H3) is a G protein-coupled receptor implicated in several disorders of the central… 
2015
2015
Histamine receptor expression in human renal tubules: a comparative pharmacological evaluation
Objective and designThe aim of this study is to evaluate the expression of the histamine receptors, particularly focusing on the… 
2015
2015
Histamine receptor expression in human renal tubules: a comparative pharmacological evaluation
The aim of this study is to evaluate the expression of the histamine receptors, particularly focusing on the H4R in human renal… 
2012
2012
Awakening properties of newly discovered highly selective H3 receptor antagonists in rats
2012
2012
A new facile synthetic route to [11C]GSK189254, a selective PET radioligand for imaging of CNS histamine H3 receptor.
2012
2012
In vivo receptor occupancy assay of histamine H₃ receptor antagonist in rats using non-radiolabeled tracer.
2009
2009
11C-GSK189254: A Selective Radioligand for In Vivo Central Nervous System Imaging of Histamine H3 Receptors by PET
The histamine H3 receptor is a G-protein–coupled presynaptic auto- and heteroreceptor whose activation leads to a decrease in the… 
Review
2007
Review
2007
Recent advances in the development of histamine H3 antagonists
The histamine H3 receptor is involved in the central and peripheral regulation of levels of histamine and other neurotransmitters… 
2006
2006
IC–P–124: Pharmacological MRI of H3 receptor antagonist GSK189254 in the rat brain
By clicking accept or continuing to use the site, you agree to the terms outlined in our Privacy Policy (opens in a new tab), Terms of Service (opens in a new tab), and Dataset License (opens in a new tab)