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Cytochrome P-450 CYP3A Inducers

Known as: Inducers, P450 CYP3A, Cytochrome P 450 CYP3A Inducers, P450 CYP3A Inducers 
Drugs and compounds that induce the synthesis of CYTOCHROME P-450 CYP3A.
National Institutes of Health

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CarbamazepineCytochrome P-450 CYP3A5 InducersNevirapinePhenobarbital
In Bloodaspects of radiation effectschemical synthesisstandards characteristics

Papers overview

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2014
2014
[Screening active components in compound danshen based on PXR-CYP3A4: an experimental study].
OBJECTIVE To screen active components in Compound Danshen (CD) based on pregnane X receptor-cytochrome P450 3A4 (PXR-CYP3A4… 
2012
2012
The Effects on Metabolic Clearance when Administering a Potent CYP3A Autoinducer with the Prototypic CYP3A Inhibitor, Ketoconazole
Ketoconazole is recognized as the prototypical CYP3A inhibitor and is often used to determine the metabolic CYP3A liabilities of… 
2005
2005
Quantitative PCR assay for cytochromes P450 2B and 3A induction in rat precision-cut liver slices: correlation study with induction in vivo.
2004
2004
GABA(A)/central benzodiazepine receptor and peripheral benzodiazepine receptor ligands as inducers of phenobarbital-inducible CYP2B and CYP3A.
2003
2003
Metabolism of medroxyprogesterone acetate (MPA) via CYP enzymes in vitro and effect of MPA on bleeding time in female rats in dependence on CYP activity in vivo.
1999
1999
Human, rat and crocodile liver microsomal monooxygenase activities measured using diazepam and nifedipine: effects of CYP3A inhibitors and relationship to immunochemically detected CYP3A apoprotein.
1999
1999
High throughput ribonuclease protection assay for the determination of CYP3A mRNA induction in cultured rat hepatocytes.
1. A rapid 96-well plate based method for the determination of CYP3A mRNA induction in primary rat hepatocytes has been developed… 
1998
1998
Strain differences in CYP3A-mediated C-8 hydroxylation (1,3,7-trimethyluric acid formation) of caffeine in Wistar and Dark Agouti rats. Rapid metabolism of caffeine in debrisoquine poor metabolizer…
1996
1996
In vivo induction of cytochrome P450 CYP3A expression in rat leukocytes using various inducers.
Highly Cited
1996
Highly Cited
1996
Cytochromes P450 (CYP) in the Poeciliopsis lucida hepatocellular carcinoma cell line (PLHC-1): dose- and time-dependent glucocorticoid potentiation of CYP1A induction without induction of CYP3A.
Glucocorticoids are being found to influence expression of cytochrome P450 (CYP) genes in multiple subfamilies in mammals (J.S… 
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