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Cyproterone

Known as: 3'H-Cyclopropa(1,2)pregna-1,4,6-triene-3,20-dione, 6-chloro-1,2-dihydro-17-hydroxy-, (1beta,2beta)-, CPTR, Cyproterone [Chemical/Ingredient] 
A synthetic steroidal anti-androgen with antineoplastic activity. Cyproterone, in its acetate form, binds the androgen receptor (AR), thereby… 
National Institutes of Health

Related topics

Related topics

14 relations

Broader (2)

Androgen Antagonistsprogesterone analog

Narrower (2)

Cyproterone AcetateSH 714
In BloodNCIt Antineoplastic Agent Terminologyagonistsanalogs & derivatives

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Highly Cited
2007
Highly Cited
2007
Modulation of steroidogenic gene expression and hormone production of H295R cells by pharmaceuticals and other environmentally active compounds.
Highly Cited
2004
Highly Cited
2004
Effects of steroid hormones on (Na+, K+)-ATPase activity inhibition-induced amnesia on the step-through passive avoidance task in gonadectomized mice.
Review
2000
Review
2000
Protocols for the Use of Cyproterone, Medroxyprogesterone, and Leuprolide in the Treatment of Paraphilia
Objective: To propose a protocol for minimizing medical complications associated with the use of cyproterone, medroxyprogesterone… 
1980
1980
Androgens inhibit estrogen action in MCF-7 human breast cancer cells.
Highly Cited
1976
Highly Cited
1976
Two sex steroid receptors in SC-115 mammary tumor cells.
Highly Cited
1975
Highly Cited
1975
Steroid-binding proteins in rabbit plasma: Separation of testosterone-binding globulin (TeBG) from corticosteroid-binding globulin (CBG), preliminary characterization of TeBG, and changes in TeBG…
1973
1973
Some biochemical effects of insulin and steroid hormones on the rat prostate in organ culture.
1972
1972
On control of spontaneous testicular regression in tree sparrows (Spizella arborea).
Highly Cited
1971
Highly Cited
1971
Distribution and metabolism of 3H-testosterone in castrated male rats; effects of cyproterone, progesterone and unlabeled testosterone.
The effect of immediate pretreatment with cyproterone, progesterone and unlabeled testosterone on the distribution and metabolism… 
Highly Cited
1969
Highly Cited
1969
Androgen Accumulation and Binding to Macromolecules in Seminal Vesicles: Inhibition by Cyproterone
Cyproterone reduces the accumulation of testosterone and dihydrotestosterone in seminal vesicles 30 minutes after intravenous… 
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