Bradykinin B2 Receptor Antagonists

Known as: Bradykinin B2 Antagonists, Antagonists, Bradykinin B2, Bradykinin B2 Receptor Inhibitors 
Compounds and drugs that inhibit ligand binding or cellular signaling by BRADYKININ B2 RECEPTORS.
National Institutes of Health

Topic mentions per year

Topic mentions per year

1991-2018
02419912018

Papers overview

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2016
2016
Bradykinin (BK) is a member of the kinin family, released in response to inflammation, trauma, burns, shock, allergy and some… (More)
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2012
2012
The bradykinin (BK) B1 receptor is an attractive target for the treatment of chronic pain and inflammation. Starting from a dual… (More)
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2009
2009
Blockade of the bradykinin B(2) receptor provides therapeutic benefit in hereditary angioedema (HAE) and potentially in many… (More)
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2002
2002
The 1-(2-nitrophenyl)thiosemicarbazide (TSC) derivative, (S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzenesulfonyl… (More)
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1999
1999
The Bradykinin B2 receptor antagonist HOE 140 (D-Arg-Arg-Pro-Hyp-Gly-Thi-Ser-D-Tic-Oic-Arg) has been used as a template for the… (More)
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Review
1999
Review
1999
Orally active nonpeptide bradykinin (BK) B2 receptor antagonists have been discovered by using directed random screening and… (More)
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1998
1998
Stimulation of the saphenous nerve in the anaesthetised rat results in cutaneous neurogenic oedema formation. We have examined… (More)
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1994
1994
1. Hoe 140, a recently described bradykinin B2 antagonist, and NPC 567 from an earlier generation of bradykinin B2 antagonists… (More)
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1992
1992
1. The effects of bradykinin on nociceptors have been characterized on a preparation of the neonatal rat spinal cord with… (More)
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1991
1991
pA2 values of new B2 receptor antagonists ranging from 7.51 to 8.86 were measured on the rabbit jugular vein, while lower values… (More)
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