Bradykinin B2 Receptor Antagonists

Known as: Bradykinin B2 Antagonists, Antagonists, Bradykinin B2, Bradykinin B2 Receptor Inhibitors 
Compounds and drugs that inhibit ligand binding or cellular signaling by BRADYKININ B2 RECEPTORS.
National Institutes of Health

Papers overview

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2009
2009
Blockade of the bradykinin B(2) receptor provides therapeutic benefit in hereditary angioedema (HAE) and potentially in many… Expand
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Highly Cited
2005
Highly Cited
2005
Pharmacological studies using bradykinin B2 receptor antagonists suggest that bradykinin, an early mediator of inflammation and… Expand
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2002
2002
The 1-(2-nitrophenyl)thiosemicarbazide (TSC) derivative, (S)-1-[4-(4-benzhydrylthiosemicarbazido)-3-nitrobenzenesulfonyl… Expand
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1999
1999
The Bradykinin B2 receptor antagonist HOE 140 (D-Arg-Arg-Pro-Hyp-Gly-Thi-Ser-D-Tic-Oic-Arg) has been used as a template for the… Expand
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Review
1999
Review
1999
Orally active nonpeptide bradykinin (BK) B2 receptor antagonists have been discovered by using directed random screening and… Expand
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1999
1999
1. Subcutaneous injection of sodium deoxycholic acid into the anterior of the back of male ddY mice elicited dose-dependent… Expand
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1998
1998
A novel class of potent, selective, and orally active non-peptide bradykinin (BK) B2 receptor antagonists were designed and… Expand
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1994
1994
1. Hoe 140, a recently described bradykinin B2 antagonist, and NPC 567 from an earlier generation of bradykinin B2 antagonists… Expand
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1992
1992
1. The effects of bradykinin on nociceptors have been characterized on a preparation of the neonatal rat spinal cord with… Expand
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1991
1991
AbstractpA2 values of new B2 receptor antagonists ranging from 7.51 to 8.86 were measured on the rabbit jugular vein, while lower… Expand
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