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Bradykinin B2 Receptor Antagonists

Known as: Bradykinin B2 Antagonists, Antagonists, Bradykinin B2, Bradykinin B2 Receptor Inhibitors 
Compounds and drugs that inhibit ligand binding or cellular signaling by BRADYKININ B2 RECEPTORS.
National Institutes of Health

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Papers overview

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2004
2004
A new series of highly potent non-peptide bradykinin B2 receptor antagonists incorporating the 4-heteroarylquinoline framework. Improvement of aqueous solubility and new insights into species…
Introduction of nitrogen-containing heteroaromatic groups at the 4-position of the quinoline moiety of our non-peptide B(2… 
1999
1999
Reduction of sodium deoxycholic acid‐induced scratching behaviour by bradykinin B2 receptor antagonists
Subcutaneous injection of sodium deoxycholic acid into the anterior of the back of male ddY mice elicited dose‐dependent… 
Review
1999
Review
1999
Discovery of orally active nonpeptide bradykinin B2 receptor antagonists.
Highly Cited
1998
Highly Cited
1998
A novel class of orally active non-peptide bradykinin B2 receptor antagonists. 3. Discovering bioisosteres of the imidazo[1,2-a] pyridine moiety.
Recently we reported on overcoming the species difference of our first orally active non-peptide bradykinin (BK) B2 receptor… 
1998
1998
Activity of tachykinin NK1 and bradykinin B2 receptor antagonists, and an opioid ligand at different stimulation parameters in neurogenic inflammation in the rat
1996
1996
Mechanisms of smokeless tobacco-induced oral mucosa inflammation: role of bradykinin.
The purpose of this study was to determine whether an aqueous extract of smokeless tobacco (moist snuff) increases clearance of… 
1996
1996
A new type of bradykinin B2 receptor antagonists: bradykinin analogs with N-alkyl amino acids at position 2.
1995
1995
Ca2+‐dependent and ‐independent mechanism of cyclic‐AMP reduction: mediation by bradykinin B2 receptors
1 Bradykinin caused a transient reduction of about 25% in the cyclic AMP level in forskolin prestimulated DDT1 MF‐2 smooth muscle… 
1995
1995
The adenylate cyclase-inhibiting bradykinin receptor in guinea pig ileum membranes exhibits an unique antagonist profile.
Highly Cited
1994
Highly Cited
1994
Agonistic and antagonistic properties of the bradykinin B2 receptor antagonist, Hoe 140, in isolated blood vessels from different species
1 Hoe 140, a recently described bradykinin B2 antagonist, and NPC 567 from an earlier generation of bradykinin B2 antagonists… 
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