Benzamidines

An iodine-catalyzed oxidative cross-coupling of C-H/N-H has been demonstrated. This simple and efficient approach constructed… Expand

Water makes it possible: The Cu(2)O-catalyzed reaction between easily available o-bromobenzylbromides and benzamidines by using… Expand

Mono-N-arylation of benzamidines 1 with aryl boronic acids 2 was effectively achieved in the presence of a catalytic amount of Cu… Expand

[RhCp*Cl(2)](2) can catalyze the oxidative coupling of N-aryl and N-alkyl benzamidines with alkynes to give N-substituted 1… Expand

A novel synthesis of 2-phenyl-4-[(triisopropylsilyl)methyl]quinazolines from monosubstituted arenes has been developed. Treatment… Expand

A series of benzamidines and benzamides was synthesized as selective inhibitors of vascular endothelial growth factor receptor… Expand

Matriptase, a trypsin-like serine protease, which may be involved in tissue remodeling, cancer invasion, and metastasis. Potent… Expand

Understanding the structural basis of inhibitor-enzyme interactions, important for the design of new drugs, requires a complete… Expand

The enzymic N-oxidation of a series of N-unsubstituted basic benzamidines (I) to a new type of metabolite, the amidoximes (II… Expand

Abstract Bovine trypsin has been purified by affinity chromatography on agarose beads containing covalently bound p… Expand