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4-azolylphenyl isoxazoline

 
National Institutes of Health

Topic mentions per year

Topic mentions per year

2002-2017
012320022017

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Isoxazoles

Related mentions per year

Related mentions per year

1946-2018
19401960198020002020
4-azolylphenyl isoxazoline
Isoxazoles

Papers overview

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2018
2018
Design, synthesis, biological evaluation and docking studies of new 3-(4,5-dihydro-1H-pyrazol/isoxazol-5-yl)-2-phenyl-1H-indole derivatives as potent antioxidants and 15-lipoxygenase inhibitors.
New candidates of 3-(4,5-dihydro-1H-pyrazol/isoxazol-5-yl)-2-phenyl-1H-indole derivatives (4-7) were designed combining the… (More)
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2017
2017
The novel isoxazoline ectoparasiticide lotilaner (Credelio™): a non-competitive antagonist specific to invertebrates γ-aminobutyric acid-gated chloride channels (GABACls)
The isoxazolines are a novel class of parasiticides that are potent inhibitors of γ-aminobutyric acid (GABA)-gated chloride… (More)
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2017
2017
NEW DRUGS IN DERMATOLOGY Prof Dr Claude FAVROT A new class of insecticides: Isoxazoline Isoxazoline is a new class of potent insecticides including Fluralaner, afoxolaner and sarolaner
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2015
2015
Discovery of an orally bioavailable isoxazoline benzoxaborole (AN8030) as a long acting animal ectoparasiticide.
A novel series of isoxazoline benzoxaborole small molecules was designed and synthesized for a structure-activity relationship… (More)
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2013
2013
4-Azolylphenyl isoxazoline insecticides acting at the GABA gated chloride channel.
Isoxazoline insecticides have been shown to be potent blockers of insect GABA receptors with excellent activity on a broad pest… (More)
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2013
2013
Inhibition by new glucocorticoid antedrugs [16α, 17α-d] isoxazoline and [16α, 17α-d]-3'-hydroxy-iminoformyl isoxazoline derivatives of chemotaxis and CCL26, CCL11, IL-8, and RANTES secretion.
The underlying inflammation present in chronic airway diseases is orchestrated by increased secretion of CC and CXC chemokines… (More)
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2009
2009
Achieving molecular complexity by organocatalytic one-pot strategies - a fast entry for synthesis of sphingoids, amino sugars, and polyhydroxylated alpha-amino acids.
A major driving force for the intriguing developments in the field of total synthesis over the past century is the proficiency… (More)
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2006
2006
Synthesis of novel 3-[5-ethyl-2-(2-phenoxy-ethyl)-pyridin]-5-substituted isoxazoline libraries via 1,3-dipolar cycloaddition and evaluation of antimicrobial activities
A series of novel 3-[5-ethyl-2-(2-phenoxy-ethyl)-pyridin]-5-substituted isoxazolines were synthesized via 1,3-dipolar… (More)
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2006
2006
In vitro anti-inflammatory activities of new steroidal antedrugs: [16alpha,17alpha-d] Isoxazoline and [16alpha,17alpha-d]-3'-hydroxy-iminoformyl isoxazoline derivatives of prednisolone and 9alpha…
A series of new anti-inflammatory steroidal antedrugs with C-16,17-isoxazoline ring system were synthesized and their… (More)
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2004
2004
Synthesis and biological evaluation of nonpeptide integrin antagonists containing spirocyclic scaffolds.
Analogues of isoxazoline alpha(v)beta(3) antagonist 1 designed to further restrict the four carbon alkyl tether were prepared by… (More)
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