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receptor antagonist activity

Interacts with receptors to reduce the action of another ligand, the agonist. [GOC:ceb, ISBN:0198506732]
National Institutes of Health

Papers overview

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2018
2018
Background Calcitonin gene-related peptide (CGRP) is a neuropeptide that acts in the trigeminovascular system and is believed to… Expand
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2015
2015
Activation of the P2X7 receptor by extracellular ATP is associated with various immune responses including allergic inflammation… Expand
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Highly Cited
2008
Highly Cited
2008
Calcium channel blockers are widely used antihypertensives. Mineralocorticoid receptor antagonists are also used to treat… Expand
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2007
2007
Type 2 diabetes is characterized by reduced insulin secretion from the pancreas and overproduction of glucose by the liver… Expand
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2004
2004
A series of novel compounds with both 5-lipoxygenase (5-LO) inhibitory and histamine H(1) receptor antagonist activity were… Expand
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1999
1999
Emesis induced by inhibitors of type IV cyclic nucleotide phosphodiesterase (PDE IV) has been investigated in the ferret. The PDE… Expand
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1993
1993
Histogranin, was co-purified with bombesin-like immunoreactive peptides from bovine adrenal medulla. Its structure, H-Met-Asn-Tyr… Expand
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1992
1992
1. The effects of the muscarinic M2 receptor antagonist methoctramine, on contractions of airway smooth muscle induced by… Expand
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1991
1991
Drugs that enhance gastrointestinal motility include the benzamide drugs metoclopramide, cisapride and renzapride (BRL-24924… Expand
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Highly Cited
1990
Highly Cited
1990
Three interleukin-1 inhibitors have been purified to homogeneity from medium conditioned by human monocytes. Partial sequence… Expand
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