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receptor antagonist activity

Interacts with receptors to reduce the action of another ligand, the agonist. [GOC:ceb, ISBN:0198506732]
National Institutes of Health

Related topics

Related topics

1 relation

Broader (1)

extracellular negative regulation of signal transduction

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2015
2015
Immunopharmacology and in fl ammation P 2 X 7 receptor antagonist activity of the anti-allergic agent oxatomide
Activation of the P2X7 receptor by extracellular ATP is associated with various immune responses including allergic inflammation… 
2010
2010
Pharmaceutical composition comprising a combination of a compound having MCHR1 antagonist activity and a compound having NPYY5 receptor antagonist activity
A compound having MCH receptor antagonist activity, a pharmaceutically acceptable salt thereof or a solvate thereof and a… 
2009
2009
Compound having npy y5 receptor antagonist activity
The present invention provides a novel compound having the compound, a pharmaceutically acceptable salt or their solvates NPY Y5… 
2000
2000
Synthesis and serotonin 2 (5-HT2) receptor antagonist activity of 5-aminoalkyl-substituted pyrrolo[3,2-c]azepines and related compounds.
A series of 5-aminoalkylpyrrolo[3,2-c]azepine derivatives was synthesized and their serotonin 2 (5-HT2) receptor antagonist and… 
2000
2000
Screening of leukotriene B4 receptor antagonist activity from the herbal drugs.
Review
1998
Review
1998
Pathophysiology and Pharmacology of Migraine. is There A Place for Antiemetics in Future Treatment Strategies?
This article reviews the pathophysiology and pharmacology of emesis in relation to migraine pathogenesis. Also, the place of… 
1994
1994
Synthesis, NMDA receptor antagonist activity, and anticonvulsant action of 1-aminocyclobutanecarboxylic acid derivatives.
A range of cis- and trans-3-substituted 1-aminocyclobutane-1-carboxylic acids has been synthesized and evaluated for antagonism… 
1993
1993
Isolation and characterization of histogranin, a natural peptide with NMDA receptor antagonist activity.
1988
1988
Leukotriene receptor antagonists. 4. Synthesis and leukotriene D4/E4 receptor antagonist activity of 4-(alkyl)acetophenone derivatives.
Analogues of the leukotriene D4/E4 receptor antagonist LY171883 (1a) were synthesized in which the tetrazole was linked to the… 
1988
1988
The thromboxane A2/prostaglandin endoperoxide receptor antagonist activity of CV-4151, a thromboxane A2 synthetase inhibitor.
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