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pravadoline

Known as: Methanone, (4-methoxyphenyl)(2-methyl-1-(2-(4-morpholinyl)ethyl)-1H-indol-3-yl)- 
National Institutes of Health

Related topics

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2 relations

Broader (1)

Indoles
pravadoline maleate

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2012
2012
Use of SPME-HS-GC-MS for the analysis of herbal products containing synthetic cannabinoids.
The increasing prevalence and use of herbal mixtures containing synthetic cannabinoids presents a growing public health concern… 
Highly Cited
1998
Highly Cited
1998
The bioactive conformation of aminoalkylindoles at the cannabinoid CB1 and CB2 receptors: insights gained from (E)- and (Z)-naphthylidene indenes.
The aminoalkylindoles (AAIs) are agonists at both the cannabinoid CB1 and CB2 receptors. To determine whether the s-trans or s… 
1998
1998
Structure-Activity Relationships of Indole-and Pyrrole-Derived Cannabinoids 1
Early molecular modeling studies with D-tetrahydrocannabinol (D-THC) reported that three discrete regions which interact with… 
1996
1996
(Aminoalkyl)indole isothiocyanates as potential electrophilic affinity ligands for the brain cannabinoid receptor.
A series of (aminoalkyl)indole compounds, naphthalene analogs of pravadoline (1), has been shown to exhibit cannabinoid agonist… 
Highly Cited
1992
Highly Cited
1992
Conformationally restrained analogues of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor.
Pravadoline (1) is an (aminoalkyl)indole analgesic agent which is an inhibitor of cyclooxygenase and, in contrast to other NSAIDs… 
Highly Cited
1992
Highly Cited
1992
Aminoalkylindole analogs: cannabimimetic activity of a class of compounds structurally distinct from delta 9-tetrahydrocannabinol.
Six novel aminoalkylindole analogs, related structurally to the dual cyclooxygenase inhibitor and nonopioid analgesic pravadoline… 
Highly Cited
1991
Highly Cited
1991
Antinociceptive (aminoalkyl)indoles.
The (aminoalkyl)indole (AAI) derivative pravadoline (1a) inhibited prostaglandin (PG) synthesis in mouse brain microsomes in… 
1990
1990
Pharmacology of pravadoline: a new analgesic agent.
Pravadoline is a new chemical entity with analgesic activity in humans. This report describes the pharmacology of pravadoline and… 
1990
1990
Pravadoline: profile in isolated tissue preparations.
Pravadoline is a novel cyclooxygenase-inhibiting analgesic with a preclinical profile of activity in vivo clearly distinct from… 
1989
1989
Pravadoline and aminoalkylindole (AAI) analogues: actions which suggest a receptor interaction.
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