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benzimidazol-2-one

National Institutes of Health

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Benzimidazoles

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2019
2019
Spiro-oxindole Piperidines and 3-(Azetidin-3-yl)-1H-benzimidazol-2-ones as mGlu2 Receptor PAMs.
Starting from two weak mGlu2 receptor positive allosteric modulator (PAM) HTS hits (4 and 5), a molecular hybridization strategy… 
2019
2019
Optimisation by Design of Experiment of Benzimidazol-2-One Synthesis under Flow Conditions
A novel flow-based approach for the preparation of benzimidazol-2-one (1) scaffold by the 1,1′-carbonyldiimidazole (CDI)-promoted… 
2010
2010
1-Isopropenyl-1H-1,3-benzimidazol-2(3H)-one
In the title N-substituted benzimidazol-2-one, C10H10N2O, the fused ring system is almost planar (r.m.s. deviation = 0.01 Å) and… 
2010
2010
Slow binding-tight binding interaction between benzimidazol-2-one inhibitors and HIV-1 reverse transcriptase containing the lysine 103 to asparagine mutation.
2009
2009
Rapid access towards follow-up NOP receptor agonists using a knowledge based approach.
2007
2007
Synthesis and evaluation of N-3 substituted phenoxypropyl piperidine benzimidazol-2-one analogues as NOP receptor agonists with analgesic and sedative properties.
2002
2002
New generation dopaminergic agents. Part 8: heterocyclic bioisosteres that exploit the 7-OH-2-(aminomethyl)chroman D(2) template.
1997
1997
Synthesis and evaluation of (S)-4-(3-(2'-[11C]isopropylamino)-2-hydroxypropoxy) -2H-benzimidazol -2-one ((S)-[11C]CGP 12388) and (S)-4-(3-((1'-[18F]-fluoroisopropyl)amino)-2-hydroxypropoxy) -2H…
The beta-adrenoceptor antagonist (S)-[11C]CGP 12177 (4-(3-(tert-butylamino)-2-hydroxypropoxy)-2H-benzimidazol -2[11C]- one) is a… 
1987
1987
Synthesis and evaluation of non-catechol D-1 and D-2 dopamine receptor agonists: benzimidazol-2-one, benzoxazol-2-one, and the highly potent benzothiazol-2-one 7-ethylamines.
Our interest in identifying D-1 and D-2 dopamine receptor agonists that are not catechols led us to extend previous studies with… 
1985
1985
1-[3-(Diarylamino)propyl]piperidines and related compounds, potential antipsychotic agents with low cataleptogenic profiles.
On the basis of a structural model of the postsynaptic dopaminergic antagonist pharmacophore, a series of 1-[3-(diarylamino… 
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