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RSR056 azetidine

National Institutes of Health

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2 relations

Broader (2)

AzetidinesPicolinic Acids

Papers overview

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2016
2016
Mechanistic interrogation of the asymmetric lithiation-trapping of N-thiopivaloyl azetidine and pyrrolidine.
A fundamental mechanistic study of the s-BuLi/chiral diamine-mediated lithiation-trapping of N-thiopivaloyl azetidine and… 
2014
2014
Nine of 16 stereoisomeric polyhydroxylated proline amides are potent β-N-acetylhexosaminidase inhibitors.
All 16 stereoisomeric N-methyl 5-(hydroxymethyl)-3,4-dihydroxyproline amides have been synthesized from lactones accessible from… 
2011
2011
Strategies to lower the Pgp efflux liability in a series of potent indole azetidine MCHR1 antagonists.
2008
2008
Stereocontrolled intramolecular cyclization of anti-β-aminonitriles. Convenient access to trans-azetidin-2-imines
We have developed a convenient approach to synthesis of trans-azetidin-2-imines, consisting in stereocontrolled cyclization of… 
2005
2005
Ccr-3 azetidine derivatives as antagonists
Formula I in free form or in salt form [Formula 1] Wherein, Ar, X, Y and T have the meanings as defined in the specification… 
2002
2002
Derives azetidine et leurs utilisations en tant qu'antagonistes de recepteur ccr3
L'invention concerne des composes de formule (I) sous forme libre ou saline, dans laquelle Ar?1, Ar2, R1?, X et n sont definis… 
2000
2000
An unexpected carbon dioxide insertion in the reaction of trans-2, 4-disubstituted azetidine, trans-2,5-disubstituted pyrrolidine, or trans-2,6-disubstituted piperidine with diphenylthiophosphinic…
In the reaction of trans-2,4-disubstituted azetidine, trans-2, 5-disubstituted pyrrolidine, or trans-2,6-disubstituted piperidine… 
2000
2000
Pharmaceutical compositions containing new or known 3-amino-azetidine derivatives having cannabinoid CB1 receptor antagonist activity, useful e.g. for treating central nervous system, respiratory or…
2000
2000
Pharmaceutical compositions containing derivatives of 3-amino-azetidine, the new derivatives and their preparation
The invention concerns pharmaceutical compositions containing as active ingredient a compound of formula (I) wherein: R1… 
1962
1962
The mechanism of the Friedel-Crafts reaction of 1-benzenesulfonyl-2-bromomethylethyleneimine with benzene
When 1-benzenesulfonyl-2-bromomethylethyleneimine, I, is treated with aluminum chloride in benzene the only identifiable product… 
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