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Endothelin A Receptor Antagonists

Known as: Antagonists, Endothelin A Receptor, Endothelin Receptor Type A Antagonist, Endothelin A Receptor Blockers 
A substance that blocks the binding of the endothelin-1 protein to its receptor. Endothelin-1 is a small molecule that causes changes in blood… 
National Institutes of Health

Papers overview

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Review
2009
Review
2009
Endothelins are a family of small peptides (ET-1, ET-2, and ET-3) that mediate various physiological processes of mitogenesis… 
Highly Cited
2002
Highly Cited
2002
The initial step of the intracellular transport of G protein-coupled receptors, their insertion into the membrane of the… 
Highly Cited
2002
Highly Cited
2002
The extracellular N terminus of the endothelin B (ETB) receptor is susceptible to limited proteolysis (cleavage at R64↓S65), but… 
Highly Cited
1998
Highly Cited
1998
The G protein β5 subunit differs substantially in amino acid sequence from the other known β subunits suggesting that βγ dimers… 
Highly Cited
1998
Highly Cited
1998
BACKGROUND Endothelin A (ETA) receptor antagonists have been shown to improve ventricular remodeling and survival in rats when… 
Highly Cited
1997
Highly Cited
1997
The endothelins (ETs) are a family of bicyclic 21-amino acid peptides that are potent and prolonged vasoconstrictors. It has been…